SCHEMBL9449128

SCHEMBL9449128

Cc1ccc(C(=O)C=[N+]=[N-])c(C)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.51
HTT P42858 4/20 0.46
ALDH1A1 P00352 4/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
HIF1A Q16665 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.40
HSD11B1 P28845 1/20 0.39
PKM P14618 2/20 0.38
ATM Q13315 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
HPGD P15428 1/20 0.38
NLRP1 Q9C000 1/20 0.38
LMNA P02545 1/20 0.38
NTSR1 P30989 1/20 0.38
FLT1 P17948 1/20 0.37
FLT4 P35916 1/20 0.37
KDR P35968 1/20 0.37
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9449019 0.83 HPGD (0.47) HTTALDH1A1KMT2AMEN1HIF1A
SCHEMBL15524099 0.83 ALDH1A1 (0.40) NFE2L2HTTALDH1A1KMT2AMEN1
SCHEMBL9449001 0.83 ALDH1A1 (0.44) NFE2L2HTTALDH1A1KMT2AMEN1
SCHEMBL15999798 0.80 ACHE (0.43) HTTALDH1A1KMT2AMEN1HIF1A
SCHEMBL28679242 0.79 HTT (0.46) NFE2L2HTTALDH1A1KMT2AMEN1
SCHEMBL11023700 0.79 NFE2L2 (0.69) NFE2L2HTTALDH1A1KMT2AMEN1
SCHEMBL11023706 0.79 NFE2L2 (0.69) NFE2L2HTTALDH1A1KMT2AMEN1
SCHEMBL9448877 0.78 GPR52 (0.45) HTTALDH1A1KMT2AMEN1HIF1A
SCHEMBL29883889 0.78 GPR52 (0.45) HTTALDH1A1KMT2AMEN1HIF1A
SCHEMBL9449020 0.77 ALDH1A1 (0.67) HTTALDH1A1KMT2AMEN1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0466730-B1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1993-07-21 EP disclosed
US-5220021-A Geminal bisphosphonic acids and derivatives as anti-arthritic agents THE UPJOHN COMPANY (US) 1993-06-15 US disclosed
WO-1990012017-A1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1990-10-18 WO disclosed