SCHEMBL9449241

SCHEMBL9449241

[N-]=[N+]=CC(=O)c1ccc(Cl)c(Cl)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
HTT P42858 1/20 0.40
HIF1A Q16665 1/20 0.40
CYP3A4 P08684 1/20 0.34
MAPK1 P28482 1/20 0.34
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GPR27 Q9NS67 1/20 0.32
MAPT P10636 1/20 0.32
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9449016 0.76 SMN1; SMN2 (0.53) ALDH1A1KMT2AMEN1HTTHIF1A
SCHEMBL9178892 0.76 MAPK1 (0.39) ALDH1A1KMT2ACYP3A4MAPK1TSHR
SCHEMBL9449288 0.76 CES2 (0.52) ALDH1A1KMT2AMEN1HTTHIF1A
SCHEMBL22123248 0.75 USP2 (0.36) ALDH1A1KMT2AMEN1HTTHIF1A
SCHEMBL15912483 0.74 FLT1 (0.41) ALDH1A1KMT2AMEN1HTTHIF1A
SCHEMBL9449019 0.74 HPGD (0.47) ALDH1A1KMT2AMEN1HTTHIF1A
SCHEMBL6787746 0.71 NPSR1 (0.44) ALDH1A1KMT2AMEN1HTTHIF1A
SCHEMBL10383925 0.70 CYP3A4 (0.34) CYP3A4MAPK1GPR27
SCHEMBL9448906 0.70 TSHR (0.52) ALDH1A1KMT2AMEN1HTTHIF1A
SCHEMBL14000033 0.70 JAK2 (0.47) ALDH1A1KMT2AMEN1HTTHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0466730-B1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1993-07-21 EP disclosed
US-5220021-A Geminal bisphosphonic acids and derivatives as anti-arthritic agents THE UPJOHN COMPANY (US) 1993-06-15 US disclosed
WO-1990012017-A1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1990-10-18 WO disclosed