SCHEMBL9449016

SCHEMBL9449016

[N-]=[N+]=CC(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.53
TSHR P16473 1/20 0.53
CASP1 P29466 1/20 0.53
ALDH1A1 P00352 4/20 0.51
MAPT P10636 4/20 0.51
MAPK1 P28482 1/20 0.49
HIF1A Q16665 1/20 0.49
RAB9A P51151 3/20 0.48
NPC1 O15118 2/20 0.48
KDM4E B2RXH2 2/20 0.47
HPGD P15428 2/20 0.44
POLB P06746 2/20 0.44
ERCC5 P28715 1/20 0.44
FEN1 P39748 1/20 0.44
SRD5A2 P31213 1/20 0.44
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HTT P42858 2/20 0.43
PKM P14618 1/20 0.43
NFKB1 P19838 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15912483 0.83 FLT1 (0.41) SMN1; SMN2TSHRCASP1ALDH1A1MAPT
SCHEMBL9449001 0.83 ALDH1A1 (0.44) SMN1; SMN2TSHRCASP1ALDH1A1MAPT
SCHEMBL9449019 0.83 HPGD (0.47) SMN1; SMN2ALDH1A1MAPTHIF1ARAB9A
SCHEMBL9448913 0.79 JAK2 (0.47) SMN1; SMN2ALDH1A1MAPTMAPK1RAB9A
SCHEMBL9449037 0.79 ABCG2 (0.49) MAPTNPC1CXCL12L3MBTL1MEN1
SCHEMBL9449288 0.78 CES2 (0.52) TSHRALDH1A1HIF1ARAB9AHPGD
SCHEMBL1697502 0.77 SMN1; SMN2 (0.61) SMN1; SMN2TSHRCASP1ALDH1A1MAPT
SCHEMBL30513965 0.77 SMN1; SMN2 (0.61) SMN1; SMN2TSHRCASP1ALDH1A1MAPT
SCHEMBL9449241 0.76 ALDH1A1 (0.40) TSHRALDH1A1MAPTMAPK1HIF1A
SCHEMBL1349424 0.76 SMN1; SMN2 (0.59) SMN1; SMN2TSHRCASP1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0466730-B1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1993-07-21 EP disclosed
US-5220021-A Geminal bisphosphonic acids and derivatives as anti-arthritic agents THE UPJOHN COMPANY (US) 1993-06-15 US disclosed
WO-1990012017-A1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1990-10-18 WO disclosed