SCHEMBL9449258

SCHEMBL9449258

CCc1cc(C#N)c(OCc2ccccc2)nc1COCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.47
SQOR Q9Y6N5 1/20 0.43
MAOB P27338 1/20 0.43
GHSR Q92847 1/20 0.40
TSHR P16473 1/20 0.39
XDH P47989 3/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
PPARG P37231 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9680846 0.80 L3MBTL1 (0.40) SQORGHSRTSHRL3MBTL1PPARG
SCHEMBL9449173 0.79 ALDH1A1 (0.44) MAOBGHSRTSHRL3MBTL1
SCHEMBL9681932 0.75 HCAR2 (0.32) CNR1TSHRPPARG
SCHEMBL30656166 0.75 CNR1 (0.54) CNR1SQORMAOB
SCHEMBL3226903 0.74 KDM4E (0.54) L3MBTL1
SCHEMBL3227733 0.74 KDM4E (0.43) CNR1XDHL3MBTL1
SCHEMBL15814214 0.71 SQOR (0.55) SQORMAOBTSHRL3MBTL1
SCHEMBL9585493 0.71 HTT (0.65)
SCHEMBL4286787 0.71 HDAC1 (0.58) CNR1SQORMAOBTSHRXDH
SCHEMBL9846090 0.71 KDM4E (0.69) TSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5202243-A Biosynthetic hydroxylation yields polymerase inhibitors MERCK & CO., INC. (US) 1993-04-13 US disclosed
US-5185251-A Treatment of HIV and AIDS MERCK & CO., INC. (US) 1993-02-09 US disclosed
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed