SCHEMBL9458418

SCHEMBL9458418

N#CC1(c2ccc(Sc3cc(C(F)(F)F)cc(C4(O)CCOCC4)c3)cc2)CCCC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 2/20 0.35
SCD O00767 1/20 0.32
NPC1 O15118 2/20 0.31
ALDH1A1 P00352 2/20 0.31
RAB9A P51151 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
SYK P43405 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
PDE2A O00408 3/20 0.31
PDE10A Q9Y233 3/20 0.31
CYP19A1 P11511 1/20 0.30
MAP4K4 O95819 1/20 0.30
OPRM1 P35372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9458637 0.82 ALOX5 (0.32) SMN1; SMN2SYKCYP19A1OPRL1
SCHEMBL9458055 0.79 WDR5 (0.34) SCDNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL9458201 0.77 OPRL1 (0.43) NPC1ALDH1A1RAB9ASMN1; SMN2SYK
SCHEMBL9458108 0.76 ALOX5 (0.34) NPC1ALDH1A1RAB9ASMN1; SMN2LMNA
SCHEMBL627580 0.71 MAP3K12 (0.44) MAP3K12SCDNPC1RAB9ATP53
SCHEMBL3158074 0.69 SLC6A3 (0.49) SCDNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL15863054 0.69 SLC6A4 (0.37) NPC1ALDH1A1RAB9ASMN1; SMN2LMNA
SCHEMBL9384364 0.69
SCHEMBL31441140 0.68 SLC6A3 (0.51) SCDNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL3516067 0.68 SLC6A3 (0.51) SCDNPC1ALDH1A1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5208259-A Lipoxygenase enzyme inhibitors IMPERIAL CHEMICAL INDUSTRIES (GB) 1993-05-04 US disclosed
EP-0409413-A2 Diaryl ether heterocycles IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-01-23 EP disclosed