SCHEMBL9467121

SCHEMBL9467121

C1=CCC(C2=CCN(CCCc3cnc4ccccc4c3)C=C2)=CC1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.32
DHODH Q02127 1/20 0.32
PDE10A Q9Y233 2/20 0.31
KDM1A O60341 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
FAAH O00519 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9719843 0.99 HTR3A (0.32) HTR3ADHODHPDE10AKDM1AMAOA
SCHEMBL9466854 0.97 HTR3A (0.32) HTR3ADHODHPDE10AKDM1AMAOA
SCHEMBL9466995 0.96 HTR3A (0.31) HTR3ADHODHPDE10AKDM1AMAOA
Hydrochloric Acid SCHEMBL9467630 0.95 HTR7 (0.31) HTR3ADHODH
SCHEMBL9466930 0.82 MGAM (0.37)
SCHEMBL8908086 0.82 ALDH1A1 (0.42) HTR3A
Water SCHEMBL9825376 0.67 LTA4H (0.37) MAOA
Hydrochloric Acid SCHEMBL9741845 0.67
SCHEMBL9825532 0.66 LTA4H (0.45)
SCHEMBL11597016 0.66 CYP1A2 (0.50) PDE10AKDM1AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5118691-A Substituted tetrahydropyridines as central nervous system agents WARNER-LAMBERT CO. (US) 1992-06-02 US claimed
US-5187280-A Dopaminergic, antipsychotic and antihypertensive agents WARNER-LAMBERT COMPANY (US) 1993-02-16 US disclosed
US-5118691-A Substituted tetrahydropyridines as central nervous system agents WARNER-LAMBERT CO. (US) 1992-06-02 US disclosed
US-5045550-A Antipsychotic, hypotensive agents, dopaminergic WARNER-LAMBERT CO. (US) 1991-09-03 US disclosed