SCHEMBL9466930

SCHEMBL9466930

O=C(CCCN1C=CC(C2=CCC=CC2)=CC1)c1cnc2ccccc2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.37
CFTR P13569 1/20 0.36
DRD2 P14416 5/20 0.35
DRD3 P35462 5/20 0.35
HTR1A P08908 3/20 0.35
HTR2A P28223 3/20 0.35
HTR2C P28335 3/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
KDM2B Q8NHM5 1/20 0.34
HDAC3 O15379 3/20 0.33
HDAC1 Q13547 3/20 0.33
ABCB1 P08183 1/20 0.31
ABCG2 Q9UNQ0 1/20 0.31
DPP4 P27487 1/20 0.31
HDAC4 P56524 2/20 0.31
HDAC7 Q8WUI4 2/20 0.31
HDAC2 Q92769 2/20 0.31
HDAC10 Q969S8 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9467121 0.82 HTR3A (0.32)
Hydrochloric Acid SCHEMBL9719843 0.81 HTR3A (0.32)
SCHEMBL9466854 0.81 HTR3A (0.32)
SCHEMBL9466995 0.81 HTR3A (0.31)
Hydrochloric Acid SCHEMBL9467630 0.80 HTR7 (0.31)
SCHEMBL8908086 0.76 ALDH1A1 (0.42) DRD2DRD3
SCHEMBL9466909 0.69 SIGMAR1 (0.58) DRD2HTR1A
SCHEMBL9360308 0.67 MGAM (0.58) MGAMCFTRHDAC3HDAC1HDAC2
SCHEMBL9631705 0.66 HTR1A (0.66) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL3382418 0.66 MGAM (0.60) MGAMCFTRHDAC3HDAC1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5118691-A Substituted tetrahydropyridines as central nervous system agents WARNER-LAMBERT CO. (US) 1992-06-02 US claimed
US-5187280-A Dopaminergic, antipsychotic and antihypertensive agents WARNER-LAMBERT COMPANY (US) 1993-02-16 US disclosed
US-5118691-A Substituted tetrahydropyridines as central nervous system agents WARNER-LAMBERT CO. (US) 1992-06-02 US disclosed
US-5045550-A Antipsychotic, hypotensive agents, dopaminergic WARNER-LAMBERT CO. (US) 1991-09-03 US disclosed