SCHEMBL9468326

SCHEMBL9468326

CC1=C(c2ccc(Cl)cc2)n2ncc(C#N)c2NC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.38
ALDH1A1 P00352 6/20 0.38
LMNA P02545 2/20 0.38
POLB P06746 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
RXRG P48443 1/20 0.37
KMT2A Q03164 5/20 0.36
HPGD P15428 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
GAA P10253 3/20 0.34
MEN1 O00255 3/20 0.34
LRRK2 Q5S007 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9478335 0.86 RXRA (0.46) KDM4EALDH1A1RXRARXRBRXRG
SCHEMBL9868786 0.76 TSHR (0.39) KDM4EALDH1A1KMT2ACNR1CNR2
SCHEMBL10554610 0.74 KDM4E (0.39) KDM4EALDH1A1LMNAPOLBRXFP1
SCHEMBL9468366 0.69 RXRA (0.39) KDM4EALDH1A1LMNAPOLBRXFP1
SCHEMBL10551237 0.64 KMO (0.36) KDM4EALDH1A1LMNAPOLBRXFP1
SCHEMBL10553556 0.63 KDM4E (0.40) KDM4EALDH1A1LMNAPOLBRXFP1
SCHEMBL10554793 0.63 RXRA (0.43) KDM4EALDH1A1RXRARXRBRXRG
SCHEMBL9870279 0.63 HTT (0.40) KMT2ANPC1RAB9A
SCHEMBL10852776 0.63 KMT2A (0.49) KDM4EALDH1A1LMNAPOLBRXFP1
SCHEMBL29157962 0.61 LRRK2 (0.34) KDM4EALDH1A1LMNAPOLBRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5219857-A Method of treating cognitive and related neural behavioral problems AMERICAN CYANAMID COMPANY (US) 1993-06-15 US disclosed
US-5126340-A Antidepressants AMERICAN CYANAMID COMPANY (US) 1992-06-30 US disclosed
US-4963553-A TREATING COGNITIVE AND NEURAL BEHAVIORAL PROBLEMS IN MAMMALS AMERICAN CYANAMID CO. (US) 1990-10-16 US disclosed