SCHEMBL9475138

SCHEMBL9475138

COc1ccc(C2C(C(=O)O)=C(C)NC(=S)N2C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.53
LMNA P02545 2/20 0.46
MAPT P10636 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
ATM Q13315 1/20 0.46
CACNA1F O60840 2/20 0.44
CACNA1D Q01668 2/20 0.44
CACNA1S Q13698 2/20 0.44
CACNA1C Q13936 2/20 0.44
KDM4E B2RXH2 4/20 0.43
GAA P10253 3/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 1/20 0.43
TP53 P04637 1/20 0.42
GUSB P08236 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
ALOX12 P18054 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9475589 0.85 KIF11 (0.53) ALDH1A1LMNAMAPTATMCACNA1F
SCHEMBL9871999 0.82 ALDH1A1 (0.47) ALDH1A1LMNAMAPTNPSR1ATM
SCHEMBL9475626 0.80 CACNA1F (0.49) ALDH1A1LMNAMAPTNPSR1CACNA1F
SCHEMBL9475421 0.78 ALDH1A1 (0.48) ALDH1A1MAPTATMCACNA1FCACNA1D
SCHEMBL9475155 0.77 ALDH1A1 (0.50) ALDH1A1ATMCACNA1FCACNA1DCACNA1S
SCHEMBL9476049 0.75 CACNA1F (0.64) ALDH1A1LMNAMAPTNPSR1CACNA1F
SCHEMBL9474962 0.74 CACNA1F (0.63) ALDH1A1LMNAMAPTNPSR1CACNA1F
SCHEMBL9475842 0.74 CACNA1F (0.47) ALDH1A1LMNAMAPTNPSR1CACNA1F
SCHEMBL9475783 0.73 LMNA (0.55) ALDH1A1LMNAMAPTCACNA1FCACNA1D
SCHEMBL27517088 0.73 KDM4E (0.68) ALDH1A1LMNAMAPTNPSR1CACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5202330-A Hypotensive and cardiovascular agent, reduces blood pressure in mammals E. R. SQUIBB & SONS, INC. (US) 1993-04-13 US disclosed
EP-0204317-A2 2-Thio or oxo-4-aryl or heterocyclo-1,5(2H)-pyrimidinedicarboxylic acid diesters and 3-acyl-5-pyrimidinecarboxylic acids and esters E.R. Squibb & Sons, Inc. (US) 1986-12-10 EP disclosed