Bromide

Bromide

SCHEMBL9475355

Br.CCOc1cc2c(cc1OCC)C(=C(C#N)SC(=N)N)NCC2

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 2/20 0.42
CHRM2 known ✓ P08172 1/20 0.42
ADRA2A known ✓ P08913 1/20 0.42
SLC6A4 known ✓ P31645 1/20 0.42
ABCC4 O15439 1/20 0.42
ABCB11 O95342 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
CHRM1 P11229 1/20 0.42
PTGS1 P23219 1/20 0.42
PDE4A P27815 1/20 0.42
KCNH2 Q12809 1/20 0.42
MAPK1 P28482 1/20 0.32
CASP1 P29466 1/20 0.32
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL9475350 1.00 ACHE (0.42) ACHEABCC4ABCB11CHRM2ADRA2A
Bromide SCHEMBL9475677 0.88 KMT2A (0.40) MAPK1CASP1KDM4EGAAMAPT
Bromide SCHEMBL9475668 0.88 KMT2A (0.40) MAPK1CASP1KDM4EGAAMAPT
Bromide SCHEMBL7430276 0.78 ACHE (0.36) ACHEPDE4AMAPK1CASP1KDM4E
Bromide SCHEMBL7433533 0.76 PDE4A (0.33) PDE4A
Bromide SCHEMBL9476998 0.75 PDPK1 (0.38) GAAMAPTHTT
SCHEMBL9475901 0.74 ACHE (0.38) ACHEABCC4ABCB11CHRM2ADRA2A
SCHEMBL9479120 0.73 ABCC4 (0.37) ACHEABCC4ABCB11CHRM2ADRA2A
Hydrochloric Acid SCHEMBL9476844 0.73 ACHE (0.37) ACHEABCC4ABCB11CHRM2ADRA2A
SCHEMBL9476362 0.73 ADRA2A (0.37) ACHEABCC4ABCB11CHRM2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5218117-A Antiallergens, antiinflammatory agents CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1993-06-08 US disclosed
US-5179089-A Antiallergens, asthma CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1993-01-12 US disclosed
EP-0486211-A1 Isoquinoline derivatives CHINOIN Gyògyszer és Vegyészeti Termékek Gyára RT. (HU) 1992-05-20 EP disclosed