SCHEMBL9476362

SCHEMBL9476362

CCOc1cc2c(cc1OCC)C(=C(C#N)SCC(O)CNC(C)(C)C)NCC2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 4/20 0.37
SLC6A4 P31645 3/20 0.37
ACHE P22303 2/20 0.37
ABCC4 O15439 1/20 0.37
ABCB11 O95342 1/20 0.37
CHRM2 P08172 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
CHRM1 P11229 1/20 0.37
PTGS1 P23219 1/20 0.37
PDE4A P27815 1/20 0.37
KCNH2 Q12809 1/20 0.37
HTR1A P08908 3/20 0.33
ADRA2B P18089 2/20 0.33
MAOA P21397 1/20 0.33
HTR2B P41595 1/20 0.33
ADRB2 P07550 4/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9477449 0.99 ADRA2A (0.36) ADRA2ASLC6A4ACHEABCC4ABCB11
SCHEMBL9475100 0.91 KMT2A (0.33) ADRA2AACHEHTR1AADRA2BMAOA
Hydrochloric Acid SCHEMBL9477098 0.90 KMT2A (0.32) ADRA2AHTR1AADRA2BMAOAHTR2B
SCHEMBL9479120 0.88 ABCC4 (0.37) ADRA2ASLC6A4ACHEABCC4ABCB11
Hydrochloric Acid SCHEMBL9477019 0.87 ABCC4 (0.37) ADRA2ASLC6A4ACHEABCC4ABCB11
SCHEMBL9475534 0.84 ADRB2 (0.36) ADRA2ASLC6A4ACHEABCC4ABCB11
Hydrochloric Acid SCHEMBL9476696 0.84 ADRB2 (0.36) ADRA2ASLC6A4ACHEABCC4ABCB11
SCHEMBL9475901 0.83 ACHE (0.38) ADRA2ASLC6A4ACHEABCC4ABCB11
Hydrochloric Acid SCHEMBL9476844 0.83 ACHE (0.37) ADRA2ASLC6A4ACHEABCC4ABCB11
SCHEMBL9476649 0.82 ABCC4 (0.37) ADRA2ASLC6A4ACHEABCC4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5179089-A Antiallergens, asthma CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1993-01-12 US claimed
EP-0486211-A1 Isoquinoline derivatives CHINOIN Gyògyszer és Vegyészeti Termékek Gyára RT. (HU) 1992-05-20 EP claimed