SCHEMBL9475534

SCHEMBL9475534

CCOc1cc2c(cc1OCC)C(=C(C#N)SCC(O)CNC1CCCCC1)NCC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.36
ABCC4 O15439 1/20 0.35
ABCB11 O95342 1/20 0.35
CHRM2 P08172 1/20 0.35
ADRA2A P08913 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
CHRM1 P11229 1/20 0.35
ACHE P22303 1/20 0.35
PTGS1 P23219 1/20 0.35
PDE4A P27815 1/20 0.35
SLC6A4 P31645 1/20 0.35
KCNH2 Q12809 1/20 0.35
LMNA P02545 1/20 0.34
KMT2A Q03164 2/20 0.32
HTR1A P08908 5/20 0.32
ADRB1 P08588 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9476696 0.99 ADRB2 (0.36) ADRB2ABCC4ABCB11CHRM2ADRA2A
SCHEMBL9476295 0.91 ADRB2 (0.35) ADRB2LMNAKMT2AKDM4EMEN1
Hydrochloric Acid SCHEMBL9476801 0.91 ADRB2 (0.35) ADRB2LMNAKMT2AKDM4EMEN1
SCHEMBL9479120 0.87 ABCC4 (0.37) ADRB2ABCC4ABCB11CHRM2ADRA2A
Hydrochloric Acid SCHEMBL9477019 0.86 ABCC4 (0.37) ADRB2ABCC4ABCB11CHRM2ADRA2A
SCHEMBL9476362 0.84 ADRA2A (0.37) ADRB2ABCC4ABCB11CHRM2ADRA2A
Hydrochloric Acid SCHEMBL9477449 0.83 ADRA2A (0.36) ADRB2ABCC4ABCB11CHRM2ADRA2A
Hydrochloric Acid SCHEMBL9476692 0.81 ABCC4 (0.36) ADRB2ABCC4ABCB11CHRM2ADRA2A
SCHEMBL9476649 0.81 ABCC4 (0.37) ADRB2ABCC4ABCB11CHRM2ADRA2A
SCHEMBL9475901 0.81 ACHE (0.38) ABCC4ABCB11CHRM2ADRA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5179089-A Antiallergens, asthma CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1993-01-12 US claimed
EP-0486211-A1 Isoquinoline derivatives CHINOIN Gyògyszer és Vegyészeti Termékek Gyára RT. (HU) 1992-05-20 EP claimed