SCHEMBL9488231

SCHEMBL9488231

C=CCC(=O)c1cccnc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLOD2 O00469 2/20 0.59
GAA P10253 2/20 0.53
ALDH1A1 P00352 2/20 0.53
APP P05067 1/20 0.53
HCAR3 P49019 1/20 0.53
HCAR2 Q8TDS4 1/20 0.53
PLOD3 O60568 1/20 0.53
PLOD1 Q02809 1/20 0.53
F7 P08709 1/20 0.52
F3 P13726 1/20 0.52
SARM1 Q6SZW1 1/20 0.52
SIRT2 Q8IXJ6 1/20 0.52
SIRT6 Q8N6T7 1/20 0.52
SIRT1 Q96EB6 1/20 0.52
SIRT3 Q9NTG7 1/20 0.52
SIRT5 Q9NXA8 1/20 0.52
SIRT4 Q9Y6E7 1/20 0.52
HDAC1 Q13547 2/20 0.49
HDAC8 Q9BY41 1/20 0.49
THRB P10828 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2693872 0.84 PLOD2 (0.61) PLOD2GAAALDH1A1APPHCAR3
SCHEMBL22978690 0.83 PLOD2 (0.56) PLOD2GAAALDH1A1APPHCAR3
SCHEMBL3982342 0.82 PLOD2 (0.59) PLOD2GAAALDH1A1APPHCAR3
SCHEMBL1583591 0.79 ALDH1A1 (0.59) PLOD2GAAALDH1A1APPHCAR3
SCHEMBL3983065 0.79 PLOD2 (0.65) PLOD2GAAALDH1A1APPHCAR3
SCHEMBL22129599 0.79 ALDH1A1 (0.53) PLOD2GAAALDH1A1APPHCAR3
SCHEMBL30633036 0.79 PLOD2 (0.51) PLOD2GAAALDH1A1APPHCAR3
SCHEMBL29145564 0.79 PLOD2 (0.51) PLOD2GAAALDH1A1APPHCAR3
SCHEMBL15662054 0.79 PLOD2 (0.51) PLOD2GAAALDH1A1APPHCAR3
SCHEMBL7075878 0.79 PLOD2 (0.69) PLOD2GAAALDH1A1APPHCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-1031768-A None JP disclosed
EP-2668161-B1 METHOD AND SUBSTANCES FOR PREPARATION OF N-SUBSTITUTED PYRIDINIUM COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 2014-11-26 EP disclosed
US-8754111-B2 Method and substances for preparation of N-substituted pyridinium compounds ROCHE DIAGNOSTICS OPERATIONS, INC. (US) 2014-06-17 US disclosed
EP-2668161-A1 METHOD AND SUBSTANCES FOR PREPARATION OF N-SUBSTITUTED PYRIDINIUM COMPOUNDS Roche Diagniostics GmbH (DE) 2013-12-04 EP disclosed
US-20130303768-A1 METHOD AND SUBSTANCES FOR PREPARATION OF N-SUBSTITUTED PYRIDINIUM COMPOUNDS ROCHE DIAGNOSTICS OPERATIONS, INC. (US) 2013-11-14 US disclosed
WO-2012101095-A1 METHOD AND SUBSTANCES FOR PREPARATION OF N-SUBSTITUTED PYRIDINIUM COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 2012-08-02 WO disclosed
EP-0302227-B1 5-HALO-6-AMINO-NICOTINIC ACID HALIDES, THEIR PREPARATION AND THEIR USE BAYER AG (DE) 1993-01-13 EP disclosed
EP-0302227-A2 5-Halo-6-amino-nicotinic acid halides, their preparation and their use BAYER AG (DE) 1989-02-08 EP disclosed
EP-0302227-A2 5-Halo-6-amino-nicotinic acid halides, their preparation and their use BAYER AG (DE) 1989-02-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130303768-A1 METHOD AND SUBSTANCES FOR PREPARATION OF N-SUBSTITUTED PYRIDINIUM COMPOUNDS PNMT, HNMT, CHRM5 PLOD2 1173/4885GAA 2997/4885ALDH1A1 870/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.