SCHEMBL949300

SCHEMBL949300

Oc1ccc(-c2ccc(O)cc2C#Cc2ccccc2)c(C#Cc2ccccc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.48
ALOX5 P09917 1/20 0.45
NPC1 O15118 2/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
RAB9A P51151 1/20 0.42
ESR2 Q92731 2/20 0.41
AKR1C2 P52895 1/20 0.41
AKR1C1 Q04828 1/20 0.41
GRM5 P41594 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6514043 0.89 ALOX5 (0.48) APPALOX5NPC1MAPTKDM4E
SCHEMBL949266 0.88 APP (0.48) APPALOX5NPC1MAPTKDM4E
SCHEMBL716896 0.84 HNF4A (0.49) APPALOX5NPC1MAPTKDM4E
SCHEMBL5049575 0.77 NPC1 (0.33) APPALOX5NPC1MAPTKDM4E
SCHEMBL4267409 0.76 APP (0.60) APPNPC1MAPTKDM4EMEN1
SCHEMBL20211704 0.76 APP (0.60) APPNPC1MAPTKDM4EMEN1
SCHEMBL11682818 0.76 MAPT (0.59) APPNPC1MAPTKDM4EMEN1
SCHEMBL5667774 0.76 TTR (0.49) APPNPC1MAPTMEN1CYP2C9
SCHEMBL6515533 0.75 HSD17B1 (0.43) APPALOX5CYP1A2CYP3A4CYP2C9
SCHEMBL717647 0.75 APP (0.67) APPNPC1MAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8519080-B2 Crosslinkable prepolymer, its production process and its uses ASAHI GLASS COMPANY, LIMITED (JP) 2013-08-27 US claimed
US-8168742-B2 Crosslinkable fluorinated aromatic prepolymer and its uses ASAHI GLASS COMPANY, LIMITED (JP) 2012-05-01 US claimed
US-9575246-B2 Prepolymer, curable material, coating composition, non-linear optical material, optical waveguide and light control device ASAHI GLASS COMPANY, LIMITED (JP) 2017-02-21 US disclosed
EP-2792665-B1 LIQUID REPELLENT COMPOSITION, LIQUID REPELLENT POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LIQUID-PHILIC REGION AND LIQUID REPELLENT REGION, AND PROCESS FOR PRODUCING IT ASAHI GLASS CO LTD (JP) 2016-08-03 EP disclosed
EP-2266792-B1 ELECTRET AND ELECTROSTATIC INDUCTION CONVERSION DEVICE ASAHI GLASS CO LTD (JP) 2016-05-04 EP disclosed
EP-2889684-A1 PREPOLYMER, CURABLE MATERIAL, COATING COMPOSITION, NON-LINEAR OPTICAL MATERIAL, OPTICAL WAVEGUIDE AND LIGHT CONTROL DEVICE Asahi Glass Company, Limited (JP) 2015-07-01 EP disclosed
US-20150153509-A1 PREPOLYMER, CURABLE MATERIAL, COATING COMPOSITION, NON-LINEAR OPTICAL MATERIAL, OPTICAL WAVEGUIDE AND LIGHT CONTROL DEVICE ASAHI GLASS COMPANY, LIMITED (JP) 2015-06-04 US disclosed
EP-2810962-A1 COMPOUND, POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LYOPHILIC REGIONS AND LYOPHOBIC REGIONS, AND METHOD FOR PRODUCING SAME Asahi Glass Company, Limited (JP) 2014-12-10 EP disclosed
EP-2792665-A1 LIQUID REPELLENT COMPOUND, LIQUID REPELLENT POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN WITH LYOPHILIC REGION AND LIQUID REPELLENT REGION, AND METHOD FOR PRODUCING SAME Asahi Glass Company, Limited (JP) 2014-10-22 EP disclosed
US-20140295149-A1 LIQUID REPELLENT COMPOSITION, LIQUID REPELLENT POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LIQUID-PHILIC REGION AND LIQUID REPELLENT REGION, AND PROCESS FOR PRODUCING IT ASAHI GLASS COMPANY, LIMITED (JP) 2014-10-02 US disclosed
US-20140287200-A1 COMPOUND, POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LIQUID-PHILIC REGION AND LIQUID REPELLENT REGION, AND PROCESS FOR PRODUCING IT ASAHI GLASS COMPANY, LIMITED (JP) 2014-09-25 US disclosed
EP-0835275-B1 IMPROVED POLY(ARYLENE ETHER) COMPOSITIONS AND THE METHOD FOR THEIR MANUFACTURE ALLIED SIGNAL INC (US) 2002-04-03 EP disclosed
US-RE37599-E1 FROM PERFLUOROBENZENE OR FLUORINATED BENZENE POLYMERS AND AROMATIC DIOLS; USE IN COATING MICROELECTRONIC STRUCTURES, SUCH AS INTEGRATED CIRCUITS; LOW DIELECTRIC CONSTANT, LOW MOISTURE ABSORPTION, AND HIGH THERMAL STABILITY. ALLIEDSIGNAL INC. 2002-03-19 US disclosed
EP-0835274-B1 PROCESS FOR MAKING HYDROXY-SUBSTITUTED ETHYNYLATED BIPHENYLS ALLIED SIGNAL INC (US) 2000-04-26 EP disclosed
US-5986045-A REACTION OF HALOARYLENE COMPOUND WITH DIPHENOL COMPOUND TO FORM POLYARYLENE ETHER ALLIEDSIGNAL INC. (US) 1999-11-16 US disclosed
US-5959157-A Process for making hydroxy-substituted ethynylated biphenyl compounds ALLIEDSIGNAL, INC. (US) 1999-09-28 US disclosed
EP-0835275-A1 IMPROVED POLY(ARYLENE ETHER) COMPOSITIONS AND THE METHOD FOR THEIR MANUFACTURE AlliedSignal Inc. (US) 1998-04-15 EP disclosed
EP-0835274-A1 HYDROXY-SUBSTITUTED ETHYNYLATED BIPHENYLS AlliedSignal Inc. (US) 1998-04-15 EP disclosed
WO-1997001593-A1 IMPROVED POLY(ARYLENE ETHER) COMPOSITIONS AND THE METHOD FOR THEIR MANUFACTURE ALLIEDSIGNAL INC. (US) 1997-01-16 WO disclosed
WO-1997001594-A1 HYDROXY-SUBSTITUTED ETHYNYLATED BIPHENYLS ALLIEDSIGNAL INC. (US) 1997-01-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140295149-A1 LIQUID REPELLENT COMPOSITION, LIQUID REPELLENT POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LIQUID-PHILIC REGION AND LIQUID REPELLENT REGION, AND PROCESS FOR PRODUCING IT CHRM1, C5, SETDB1 APP 1777/4885ALOX5 1117/4885NPC1 1372/4885
US-20140287200-A1 COMPOUND, POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LIQUID-PHILIC REGION AND LIQUID REPELLENT REGION, AND PROCESS FOR PRODUCING IT H1-0, DNMT1, BMI1 APP 1763/4885ALOX5 3276/4885NPC1 1590/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.