SCHEMBL9494728

SCHEMBL9494728

CN(C(=O)Cc1cccc2ccccc12)C1c2ccccc2CCC1N1CCCC1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.67
OPRM1 P35372 9/20 0.64
OPRK1 P41145 9/20 0.64
OPRD1 P41143 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9702348 0.96 SIGMAR1 (0.67) SIGMAR1OPRM1OPRK1OPRD1
SCHEMBL9767727 0.90 SIGMAR1 (0.66) SIGMAR1OPRM1OPRK1OPRD1
Hydrochloric Acid SCHEMBL9767758 0.89 SIGMAR1 (0.65) SIGMAR1OPRM1OPRK1OPRD1
SCHEMBL9702542 0.87 OPRM1 (0.66) SIGMAR1OPRM1OPRK1OPRD1
SCHEMBL10589759 0.83 SIGMAR1 (0.76) SIGMAR1OPRM1OPRK1OPRD1
SCHEMBL9703418 0.83 OPRM1 (0.66) SIGMAR1OPRM1OPRK1OPRD1
SCHEMBL10588635 0.79 SIGMAR1 (0.70) SIGMAR1OPRM1OPRK1OPRD1
SCHEMBL9494140 0.79 SIGMAR1 (0.51) SIGMAR1OPRM1OPRK1OPRD1
SCHEMBL9748668 0.78 OPRK1 (1.00) SIGMAR1OPRM1OPRK1OPRD1
SCHEMBL9748062 0.78 OPRK1 (1.00) SIGMAR1OPRM1OPRK1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0329563-B1 BENZOCYCLOHEXANE AND BENZOCYCLOHEPTANE DERIVATIVES AND THEIR SALTS, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, THEIR USE AS MEDICINES AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-04-21 EP claimed
US-5130329-A Amino, amide substituted compounds ROUSSEL UCLAF (FR) 1992-07-14 US disclosed
US-5068244-A Benzcarbocyclic amides with nitro groups ROUSSEL UCLAF (FR) 1991-11-26 US disclosed