SCHEMBL9494140

SCHEMBL9494140

O=C(Cc1cccc2ccccc12)NC1c2ccccc2CCC1N1CCCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.51
OPRM1 P35372 2/20 0.48
OPRK1 P41145 2/20 0.48
ALDH1A1 P00352 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 3/20 0.44
PREP P48147 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
MAPT P10636 1/20 0.43
GSK3B P49841 1/20 0.42
CDK5 Q00535 1/20 0.42
CDK5R1 Q15078 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
NCOR2 Q9Y618 1/20 0.42
LMNA P02545 1/20 0.41
HPGD P15428 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9493289 0.96 SIGMAR1 (0.51) SIGMAR1OPRM1OPRK1ALDH1A1SMN1; SMN2
SCHEMBL9493356 0.85 OPRM1 (0.69) OPRM1OPRK1
SCHEMBL9494197 0.81 OPRM1 (0.69) OPRM1OPRK1
SCHEMBL9494728 0.79 SIGMAR1 (0.67) SIGMAR1OPRM1OPRK1OPRD1
SCHEMBL9493563 0.76 SIGMAR1 (0.50) SIGMAR1OPRM1OPRK1ALDH1A1SMN1; SMN2
SCHEMBL9702348 0.75 SIGMAR1 (0.67) SIGMAR1OPRM1OPRK1OPRD1
SCHEMBL9493252 0.72 OPRD1 (0.52) SIGMAR1ALDH1A1HDAC3HDAC1HDAC8
SCHEMBL9496739 0.71 ALDH1A1 (0.53) SIGMAR1ALDH1A1SMN1; SMN2KDM4EMEN1
SCHEMBL7628560 0.71 MTNR1A (0.46) OPRM1OPRK1ALDH1A1SMN1; SMN2
SCHEMBL7628567 0.71 MTNR1A (0.46) OPRM1OPRK1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0329563-B1 BENZOCYCLOHEXANE AND BENZOCYCLOHEPTANE DERIVATIVES AND THEIR SALTS, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, THEIR USE AS MEDICINES AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-04-21 EP claimed
EP-0329563-A2 Benzocyclohexane and benzocycloheptane derivatives and their salts, process and intermediates for their preparation, their use as medicines and compositions containing them ROUSSEL-UCLAF (FR) 1989-08-23 EP claimed
EP-0329563-B1 BENZOCYCLOHEXANE AND BENZOCYCLOHEPTANE DERIVATIVES AND THEIR SALTS, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, THEIR USE AS MEDICINES AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-04-21 EP disclosed
EP-0329563-A2 Benzocyclohexane and benzocycloheptane derivatives and their salts, process and intermediates for their preparation, their use as medicines and compositions containing them ROUSSEL-UCLAF (FR) 1989-08-23 EP disclosed