SCHEMBL9502663

SCHEMBL9502663

O=C(OC(C(=O)NCc1ccccc1)c1ccccc1)c1cccnc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.55
KMT2A Q03164 5/20 0.54
LMNA P02545 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
HTT P42858 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
HPGD P15428 1/20 0.51
GAA P10253 1/20 0.51
BCHE P06276 1/20 0.50
SLC1A2 P43004 1/20 0.50
KLK7 P49862 1/20 0.49
ALDH1A1 P00352 2/20 0.48
PKM P14618 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
EPHX2 P34913 1/20 0.48
CYP3A4 P08684 1/20 0.47
TSHR P16473 1/20 0.47
MEN1 O00255 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9503442 0.87 CYP2D6 (0.66) CYP2D6KMT2ALMNAKLK7ALDH1A1
SCHEMBL28924092 0.81 ALDH1A1 (0.53) KMT2ALMNATDP1HTTGAA
SCHEMBL11630201 0.81 ALDH1A1 (0.53) KMT2ALMNATDP1HTTGAA
Niacin SCHEMBL9502658 0.78 SMN1; SMN2 (0.53) KMT2ALMNAHTTSMN1; SMN2HPGD
SCHEMBL4158522 0.75 PKM (0.62) KMT2ALMNAHTTKLK7ALDH1A1
SCHEMBL4162007 0.75 PKM (0.62) KMT2ALMNAHTTKLK7ALDH1A1
SCHEMBL4158526 0.75 PKM (0.62) KMT2ALMNAHTTKLK7ALDH1A1
SCHEMBL354041 0.75 TSHR (0.76) KMT2ASMN1; SMN2GAAL3MBTL1CYP2C9
SCHEMBL9478771 0.75 ESR1 (0.57) KMT2ALMNATDP1HTTGAA
Iodide SCHEMBL15903217 0.74 TSHR (0.74) KMT2ASMN1; SMN2GAACYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0376852-B1 MICROGRANULES ESSENTIALLY CONSISTING OF TRIGLYCERIDES OF SATURATED FATTY ACIDS LOADED WITH AN ACTIVE SUBSTANCE, AND THEIR TOPICAL THERAPEUTICAL USE CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA - CIRD GALDERMA (FR) 1993-06-23 EP claimed