SCHEMBL9504458

SCHEMBL9504458

CCCN(CCOc1c(Cl)cccc1Cl)C1Cc2cc(O)c(O)cc2C1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FYN P06241 2/20 0.62
DRD3 P35462 9/20 0.48
DRD2 P14416 8/20 0.48
DRD4 P21917 5/20 0.46
CYP2D6 P10635 2/20 0.46
HTR1A P08908 2/20 0.46
MEN1 O00255 2/20 0.46
ADRB2 P07550 2/20 0.46
KMT2A Q03164 2/20 0.46
CASP1 P29466 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP2C9 P11712 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
LMNA P02545 2/20 0.45
DRD1 P21728 1/20 0.45
DRD5 P21918 1/20 0.45
HTR7 P34969 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9503275 0.91 FYN (0.58) FYNDRD3DRD2DRD4CYP2D6
SCHEMBL9507046 0.85 DRD2 (0.55) FYNDRD3DRD2DRD4HTR1A
SCHEMBL9507115 0.81 DRD2 (0.70) DRD3DRD2DRD4HTR1AADRB2
Hydrochloric Acid SCHEMBL9504453 0.80 DRD2 (0.69) DRD3DRD2DRD4HTR1AADRB2
SCHEMBL9504552 0.79 DRD2 (0.61) DRD3DRD2DRD4HTR1AADRB2
SCHEMBL8443814 0.79 FYN (1.00) FYNDRD3DRD2DRD4CYP2D6
Bromide SCHEMBL8689149 0.77 FYN (0.96) FYNDRD3DRD2DRD4CYP2D6
SCHEMBL9504450 0.76 DRD2 (0.54) DRD3DRD2DRD4CYP2D6HTR1A
Hydrochloric Acid SCHEMBL9507124 0.75 DRD2 (0.55) DRD3DRD2DRD4CYP2D6HTR1A
SCHEMBL9503307 0.73 ADRA2A (0.48) FYNDRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0321968-B1 COMPOUNDS ACTIVE ON THE CARDIOVASCULAR SYSTEM ZAMBON GROUP S.p.A. (IT) 1993-07-28 EP disclosed
US-5151414-A Hypotensive agents SIMES SOCIETA ITALIANA MEDICINALI E SINTETICI S.P.A. (IT) 1992-09-29 US disclosed
US-5070106-A HYPOTENSIVES, CEREBRAL DISORDERS SIMES SOCIETA ITALIANA MEDICINALI E SINTETICI S.P.A. (IT) 1991-12-03 US disclosed