SCHEMBL9505019

SCHEMBL9505019

CCc1cc(C(F)(F)F)nc(N(C(N)=O)c2ccccc2[N+](=O)[O-])n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
GAA P10253 1/20 0.35
P2RX1 P51575 2/20 0.34
IGF1R P08069 1/20 0.34
KMT2A Q03164 5/20 0.33
MEN1 O00255 4/20 0.33
MAPT P10636 4/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
ALDH1A1 P00352 4/20 0.33
POLB P06746 1/20 0.33
CES2 O00748 1/20 0.33
ACHE P22303 1/20 0.33
CES1 P23141 1/20 0.33
HTT P42858 2/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9504996 0.85 CYP1A2 (0.37) CYP1A2CYP3A4CYP2C19GAAP2RX1
SCHEMBL9818596 0.78 MEN1 (0.36) CYP1A2CYP3A4CYP2C19GAAP2RX1
SCHEMBL9738579 0.76 PRKD3 (0.43)
SCHEMBL9739910 0.76 PDE4B (0.35) CYP3A4CYP2C19GAAIGF1RKMT2A
SCHEMBL10400918 0.75 ALDH1A1 (0.35) CYP1A2CYP3A4CYP2C19GAAKMT2A
SCHEMBL9539862 0.74 ALDH1A1 (0.35) P2RX1KMT2AMEN1PDK1PDK2
SCHEMBL10517413 0.73 ALDH1A1 (0.34) CYP1A2CYP3A4CYP2C19P2RX1KMT2A
SCHEMBL9818604 0.72 NPC1 (0.43) KMT2AMEN1ALDH1A1POLBNPC1
SCHEMBL10400826 0.72 F2 (0.34) P2RX1KMT2AMEN1MAPTPDK1
SCHEMBL10458605 0.72 KMT2A (0.40) CYP1A2CYP2C19KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337946-B1 UREAS CIBA-GEIGY AG (CH) 1993-07-28 EP claimed
US-4999046-A Herbicides and plant growth regulators, agricultural use CIBA-GEIGY CORPORATION (US) 1991-03-12 US claimed
EP-0337946-A1 Ureas CIBA-GEIGY AG (CH) 1989-10-18 EP claimed
EP-0337946-B1 UREAS CIBA-GEIGY AG (CH) 1993-07-28 EP disclosed
US-4999046-A Herbicides and plant growth regulators, agricultural use CIBA-GEIGY CORPORATION (US) 1991-03-12 US disclosed
EP-0337946-A1 Ureas CIBA-GEIGY AG (CH) 1989-10-18 EP disclosed