SCHEMBL9539862

SCHEMBL9539862

Cc1c(Cl)nc(N(C(N)=O)c2ccccc2[N+](=O)[O-])nc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
TAS1R2 Q8TE23 1/20 0.34
HTT P42858 1/20 0.33
ATM Q13315 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
P2RX1 P51575 1/20 0.33
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
POLB P06746 2/20 0.32
CYP2C9 P11712 1/20 0.32
DHODH Q02127 1/20 0.32
LMNA P02545 2/20 0.32
TSHR P16473 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10400826 0.87 F2 (0.34) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL10517413 0.86 ALDH1A1 (0.34) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL10400918 0.83 ALDH1A1 (0.35) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL10400124 0.82 LMNA (0.34) ALDH1A1TAS1R3TAS1R1TAS1R2HTT
SCHEMBL10400122 0.81 TAS1R3 (0.34) ALDH1A1TAS1R3TAS1R1TAS1R2HTT
SCHEMBL9536988 0.78 SMN1; SMN2 (0.37) ALDH1A1SMN1; SMN2P2RX1MEN1KMT2A
SCHEMBL9536239 0.78 SMN1; SMN2 (0.35) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL9535151 0.77 LMNA (0.34) ALDH1A1TAS1R3TAS1R1TAS1R2HTT
SCHEMBL10458605 0.77 KMT2A (0.40) ALDH1A1HTTATMSMN1; SMN2MEN1
SCHEMBL10400150 0.77 MAPK14 (0.41) PDK1PDK2PDK3PDK4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337944-B1 UREAS CIBA-GEIGY AG (CH) 1993-07-28 EP disclosed
US-4973690-A PYRIMIDIN-2-YL UREAS, HERBICICES, PLANT GROWTH REGULATORS CIBA-GEIGY CORPORATION (US) 1990-11-27 US disclosed
EP-0337944-A1 Ureas CIBA-GEIGY AG (CH) 1989-10-18 EP disclosed