SCHEMBL9064752

SCHEMBL9064752

C=CCOC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.74
ALDH1A1 P00352 4/20 0.71
KDM4E B2RXH2 3/20 0.71
HSD17B10 Q99714 2/20 0.71
TP53 P04637 2/20 0.71
HPGD P15428 2/20 0.71
CACNA1D Q01668 4/20 0.68
CACNA1F O60840 3/20 0.68
CACNA1S Q13698 3/20 0.68
CACNA1C Q13936 3/20 0.68
MAPT P10636 3/20 0.63
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
LMNA P02545 1/20 0.63
GAA P10253 1/20 0.63
MAPK1 P28482 1/20 0.63
CACNA1B Q00975 2/20 0.62
CA1 P00915 1/20 0.62
CA2 P00918 1/20 0.62
POLB P06746 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10475395 0.95 ALDH1A1 (0.78) ADORA3ALDH1A1KDM4EHSD17B10TP53
SCHEMBL10475396 0.91 CACNA1B (0.74) ADORA3ALDH1A1KDM4EHSD17B10TP53
SCHEMBL24469031 0.90 ALDH1A1 (0.68) ADORA3ALDH1A1KDM4EHSD17B10TP53
SCHEMBL9505249 0.87 ALDH1A1 (0.67) ADORA3ALDH1A1KDM4EHSD17B10TP53
SCHEMBL20610477 0.85 ADORA3 (1.00) ADORA3ALDH1A1KDM4EHSD17B10TP53
SCHEMBL3905675 0.85 ADORA3 (0.83) ADORA3ALDH1A1KDM4EHSD17B10TP53
SCHEMBL4935843 0.84 KDM4E (0.82) ADORA3ALDH1A1KDM4EHSD17B10TP53
SCHEMBL11776554 0.83 KDM4E (0.56) ADORA3ALDH1A1KDM4EHSD17B10TP53
SCHEMBL10732135 0.83 MAPT (0.64) ADORA3ALDH1A1KDM4EHSD17B10TP53
SCHEMBL9502940 0.83 MEN1 (0.79) ADORA3CACNA1DCACNA1FCACNA1SCACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996033972-A1 METHODS FOR SYNTHESIZING DIVERSE COLLECTIONS OF PYRIDINES, PYRIMIDINES, 1,4-DIHYDRO DERIVATIVES THEREOF, AND PIPERIDINE DERIVATIVES GLAXO GROUP LIMITED (GB) 1996-10-31 WO disclosed