SCHEMBL9505703

SCHEMBL9505703

COCc1cc(C)nc(Nc2ccccc2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.54
SMN1; SMN2 Q16637 4/20 0.50
KCNH3 Q9ULD8 2/20 0.50
HTT P42858 2/20 0.50
VSIR Q9H7M9 1/20 0.49
KDM4E B2RXH2 3/20 0.47
MAPT P10636 3/20 0.47
LMNA P02545 1/20 0.47
GPR55 Q9Y2T6 1/20 0.47
MEN1 O00255 1/20 0.46
HPGD P15428 1/20 0.46
KMT2A Q03164 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
KCNH2 Q12809 1/20 0.45
ALDH1A1 P00352 1/20 0.44
USP2 O75604 1/20 0.44
POLB P06746 1/20 0.44
ALOX15 P16050 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9505657 0.85 RAB9A (0.48) HTTKDM4EMAPTLMNAMEN1
SCHEMBL13547969 0.85 KCNH3 (0.50) TAAR1SMN1; SMN2KCNH3HTTVSIR
SCHEMBL13547970 0.84 VSIR (0.51) SMN1; SMN2KCNH3HTTVSIRMAPT
SCHEMBL9763194 0.81 TAAR1 (0.56) TAAR1SMN1; SMN2HTTKDM4EMAPT
SCHEMBL9762820 0.81 TAAR1 (0.56) TAAR1SMN1; SMN2KCNH3HTTVSIR
SCHEMBL9762436 0.81 TAAR1 (0.47) TAAR1SMN1; SMN2KCNH3HTTVSIR
SCHEMBL9502856 0.80 KCNH3 (0.46) SMN1; SMN2KCNH3VSIRMAPTMEN1
Pyrimethanil SCHEMBL20817 0.80 SMN1; SMN2 (0.71) TAAR1SMN1; SMN2KCNH3HTTKDM4E
SCHEMBL27261700 0.79 TAAR1 (0.54) TAAR1SMN1; SMN2KCNH3HTTKDM4E
SCHEMBL2206867 0.79 MAPT (0.43) TAAR1SMN1; SMN2KCNH3HTTVSIR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0295210-B1 MICROBICIDES CIBA-GEIGY AG (CH) 1993-08-04 EP claimed
EP-0295210-A1 Microbicides CIBA-GEIGY AG (CH) 1988-12-14 EP claimed
US-9006243-B2 HIV inhibiting 6-substituted pyrimidines JANSSEN R&D IRELAND (IE) 2015-04-14 US disclosed
US-20100016317-A1 HIV INHIBITING 6-SUBSTITUTED PYRIMIDINES JANSSEN SCIENCES IRELAND UC (IE) 2010-01-21 US disclosed
EP-0295210-B1 MICROBICIDES CIBA-GEIGY AG (CH) 1993-08-04 EP disclosed
EP-0270111-B1 PYRIMIDINE DERIVATIVES AND AGRICULTURAL OR HORTICULTURAL FUNGICIDAL COMPOSITION CONTANING THE SAME KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1991-05-15 EP disclosed
US-4992438-A Pyrimidine derivatives, process for preparing the same and agricultural or horticultural fungicidal composition containing the same KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1991-02-12 US disclosed
US-4897396-A AGRICULTURAL INSECTICIDES, PESTICIDES AND FUNGICIDES CIBA-GEIGY CORPORATION (US) 1990-01-30 US disclosed
EP-0295210-A1 Microbicides CIBA-GEIGY AG (CH) 1988-12-14 EP disclosed
EP-0270111-A1 Pyrimidine derivatives and agricultural or horticultural fungicidal composition contaning the same KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1988-06-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100016317-A1 HIV INHIBITING 6-SUBSTITUTED PYRIMIDINES CCR5, CTR9, NR1H3 TAAR1 2495/4885SMN1; SMN2 4738/4885KCNH3 1012/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.