SCHEMBL9506940

SCHEMBL9506940

O=C(O)CCCCCC(c1ccc(F)cc1)c1cc(Br)c2ccccc2c1O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 4/20 0.53
TBXAS1 P24557 1/20 0.41
RCE1 Q9Y256 1/20 0.41
KCNH2 Q12809 2/20 0.37
SLC6A3 Q01959 4/20 0.36
CACNA1F O60840 2/20 0.36
DRD4 P21917 2/20 0.36
DRD5 P21918 2/20 0.36
HRH2 P25021 2/20 0.36
ADRA1D P25100 2/20 0.36
HTR2A P28223 2/20 0.36
HTR7 P34969 2/20 0.36
ADRA1A P35348 2/20 0.36
HRH1 P35367 2/20 0.36
ADRA1B P35368 2/20 0.36
OPRM1 P35372 2/20 0.36
DRD3 P35462 2/20 0.36
OPRD1 P41143 2/20 0.36
OPRK1 P41145 2/20 0.36
HTR6 P50406 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9510689 0.83 TBXA2R (0.56) TBXA2RTBXAS1RCE1
SCHEMBL67664 0.75 TBXA2R (0.65) TBXA2RTBXAS1SLC6A3CACNA1FDRD4
SCHEMBL9699510 0.70 TBXA2R (0.82) TBXA2RTBXAS1KCNH2SLC6A3
SCHEMBL67079 0.70 TBXA2R (0.58) TBXA2RTBXAS1SLC6A3CACNA1FDRD4
SCHEMBL8742992 0.69 TBXA2R (0.58) TBXA2RLTB4R
SCHEMBL8743003 0.69 TBXA2R (0.58) TBXA2RLTB4R
SCHEMBL8743193 0.69 TBXA2R (0.76) TBXA2RTBXAS1KCNH2SLC6A3HTR2A
SCHEMBL9507218 0.69 TBXA2R (0.76) TBXA2RTBXAS1KCNH2SLC6A3HTR2A
SCHEMBL8743182 0.69 TBXA2R (0.76) TBXA2RTBXAS1KCNH2SLC6A3HTR2A
SCHEMBL7683666 0.69 TBXAS1 (0.73) TBXA2RTBXAS1SLC6A3HTR2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0295037-B1 PHENOL DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-08-18 EP disclosed
US-5162571-A Phenol derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-11-10 US disclosed
EP-0295037-A2 Phenol derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1988-12-14 EP disclosed