SCHEMBL9508027

SCHEMBL9508027

COc1cc(C(=O)CCCCCBr)cc(C(C)C)c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.42
POLB P06746 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
THPO P40225 1/20 0.41
MTOR P42345 1/20 0.41
PMP22 Q01453 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5841291 0.86 MEN1 (0.53) MAPK1POLBSMN1; SMN2KMT2AMEN1
SCHEMBL24722331 0.76 MEN1 (0.55) MAPK1POLBSMN1; SMN2KMT2AMEN1
SCHEMBL5355533 0.75 CTNNB1 (0.63) POLBSMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL11042463 0.75 MEN1 (0.51) MAPK1POLBSMN1; SMN2KMT2AMEN1
SCHEMBL27200216 0.75 CTNNB1 (0.63) POLBSMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL7834034 0.74 MEN1 (0.56) MAPK1POLBSMN1; SMN2KMT2AMEN1
SCHEMBL23534095 0.73 POLB (0.41) MAPK1POLBSMN1; SMN2KMT2AMEN1
SCHEMBL29767827 0.73 POLB (0.41) MAPK1POLBSMN1; SMN2KMT2AMEN1
SCHEMBL9828028 0.73 MEN1 (0.62) MAPK1POLBSMN1; SMN2KMT2AMEN1
SCHEMBL9119840 0.73 CTNNB1 (0.65) POLBSMN1; SMN2KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0310126-B1 DERIVATIVES OF PYROCATECHOL-CARBOXYLIC ACID, THEIR PREPARATION AND USE AS ACTIVE INGREDIENTS IN MEDICINES F. HOFFMANN-LA ROCHE AG (CH) 1993-08-18 EP disclosed
US-5191108-A Lipoxygenase inhibitors, antiinflammatory agents HOFFMANN-LA ROCHE INC. (US) 1993-03-02 US disclosed
US-5025036-A Antiinflammatory agents, gastrointestinal, cardiovascular and skin disorders HOFFMANN-LA ROCHE INC. (US) 1991-06-18 US disclosed
US-4937373-A Substituted naphthalene carboxylic acids HOFFMANN-LA ROCHE INC. (US) 1990-06-26 US disclosed
EP-0310126-A2 Derivatives of pyrocatechol-carboxylic acid, their preparation and use as active ingredients in medicines F. HOFFMANN-LA ROCHE AG (CH) 1989-04-05 EP disclosed