SCHEMBL9508313

SCHEMBL9508313

FC(F)(F)C1(c2ccccc2)CCCc2ccc(Cl)cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.46
SIGMAR1 Q99720 6/20 0.40
PDK2 Q15119 4/20 0.40
MAP3K14 Q99558 1/20 0.36
HTR2A P28223 3/20 0.34
HTR2C P28335 3/20 0.34
DRD2 P14416 2/20 0.34
HTR2B P41595 2/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
DRD1 P21728 1/20 0.34
ADRA1A P35348 1/20 0.34
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9509084 0.90 SIGMAR1 (0.48) KDM1ASIGMAR1PDK2MAP3K14SLC6A4
SCHEMBL9509061 0.84 SIGMAR1 (0.46) KDM1ASIGMAR1PDK2HTR2AHTR2C
SCHEMBL9511025 0.83 KIF11 (0.40) KDM1ASIGMAR1PDK2HTR2AHTR2C
SCHEMBL9509760 0.83 KDM1A (0.42) KDM1ASIGMAR1HTR2AHTR2CDRD2
SCHEMBL9509089 0.82 PDK2 (0.40) KDM1ASIGMAR1PDK2AKR1B1
SCHEMBL9508316 0.79 SIGMAR1 (0.50) KDM1ASIGMAR1PDK2DRD2DRD1
SCHEMBL24275635 0.75 KDM1A (0.50) KDM1ASIGMAR1PDK2HTR2AHTR2C
SCHEMBL9509096 0.74 KDM1A (0.49) KDM1APDK2
SCHEMBL9509759 0.73 KDM1A (0.40) KDM1ASIGMAR1PDK2HTR2AHTR2C
SCHEMBL24275641 0.71 KDM1A (0.56) KDM1ASIGMAR1PDK2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0414686-B1 DERIVATIVES OF TRIFLUOROMETHYL-1-TETRALINES, PREPARATION AND APPLICATION THEREOF FOR THE SYNTHESIS OF COMPOUNDS HAVING THERAPEUTIC PROPERTIES LABORATOIRES LUCIEN (FR) 1993-09-22 EP claimed