SCHEMBL9509760

SCHEMBL9509760

FC(F)(F)C1(c2ccccc2)CCCc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 3/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
SIGMAR1 Q99720 8/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
DRD2 P14416 1/20 0.40
TSHR P16473 1/20 0.40
NFKB1 P19838 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTR2B P41595 1/20 0.40
MTOR P42345 1/20 0.40
AKR1B1 P15121 1/20 0.40
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9509061 0.87 SIGMAR1 (0.46) KDM1AMEN1KMT2ASIGMAR1TP53
SCHEMBL9511025 0.84 KIF11 (0.40) KDM1AMEN1KMT2ASIGMAR1TP53
SCHEMBL9508294 0.84 SIGMAR1 (0.48) KDM1AMEN1KMT2ASIGMAR1DRD2
SCHEMBL9509089 0.83 PDK2 (0.40) KDM1ASIGMAR1AKR1B1
SCHEMBL9508313 0.83 KDM1A (0.46) KDM1ASIGMAR1TP53CYP1A2CYP3A4
SCHEMBL9509759 0.82 KDM1A (0.40) KDM1AMEN1KMT2ASIGMAR1TP53
SCHEMBL9509084 0.82 SIGMAR1 (0.48) KDM1ASIGMAR1
SCHEMBL9512045 0.80 SIGMAR1 (0.43) KDM1AMEN1KMT2ASIGMAR1DRD2
SCHEMBL9508316 0.79 SIGMAR1 (0.50) KDM1ASIGMAR1DRD2
SCHEMBL9509137 0.79 MEN1 (0.42) KDM1AMEN1KMT2ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0414686-B1 DERIVATIVES OF TRIFLUOROMETHYL-1-TETRALINES, PREPARATION AND APPLICATION THEREOF FOR THE SYNTHESIS OF COMPOUNDS HAVING THERAPEUTIC PROPERTIES LABORATOIRES LUCIEN (FR) 1993-09-22 EP claimed
US-5091429-A Antidepressant and analgesic with side effects reduction LABORATOIRES LUCIEN (FR) 1992-02-25 US disclosed