SCHEMBL9508502

SCHEMBL9508502

CC(C)CC1c2ccccc2CCN1C(=O)C(Cl)Cl

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 4/20 0.57
ACE P12821 2/20 0.49
HHAT Q5VTY9 3/20 0.48
DRD1 P21728 1/20 0.47
CYP2D6 P10635 5/20 0.45
NPSR1 Q6W5P4 1/20 0.44
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
MTNR1A P48039 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9509872 0.87 MTNR1B (0.53) MTNR1BACEHHATDRD1CYP2D6
SCHEMBL9509163 0.85 MTNR1B (0.51) MTNR1BACEHHATDRD1NPSR1
SCHEMBL9508177 0.80 ACE (0.49) MTNR1BACEHHATDRD1CYP2D6
SCHEMBL2138396 0.80 DRD1 (0.59) MTNR1BACEHHATDRD1CYP2D6
SCHEMBL10770517 0.79 ACE (0.48) MTNR1BACEHHATDRD1CYP2D6
SCHEMBL9511054 0.76 ACE (0.45) MTNR1BACEHHATDRD1CYP2D6
SCHEMBL19010155 0.75 PRCP (0.51) MTNR1BDRD1OPRM1OPRD1
SCHEMBL19010161 0.75 PRCP (0.51) MTNR1BDRD1OPRM1OPRD1
SCHEMBL19010148 0.75 PRCP (0.51) MTNR1BDRD1OPRM1OPRD1
SCHEMBL9508456 0.75 HHAT (0.57) HHATCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0230871-B1 HALOACYL 1-SUBSTITUTED-1,2,3,4-TETRAHYDROISOQUINOLINES AS HERBICIDE ANTIDOTES Monsanto Company (US) 1993-09-22 EP claimed
EP-0230871-A2 Haloacyl 1-substituted-1,2,3,4-tetrahydroisoquinolines as herbicide antidotes Monsanto Company (US) 1987-08-05 EP claimed
EP-0230871-B1 HALOACYL 1-SUBSTITUTED-1,2,3,4-TETRAHYDROISOQUINOLINES AS HERBICIDE ANTIDOTES Monsanto Company (US) 1993-09-22 EP disclosed
US-4755218-A Reducing acetochlor injury to corn by applying with antidote MONSANTO COMPANY (US) 1988-07-05 US disclosed
EP-0230871-A2 Haloacyl 1-substituted-1,2,3,4-tetrahydroisoquinolines as herbicide antidotes Monsanto Company (US) 1987-08-05 EP disclosed