SCHEMBL9511054

SCHEMBL9511054

CC(C)(C)C1c2ccccc2CCN1C(=O)C(Cl)Cl

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACE P12821 4/20 0.45
MTNR1B P49286 1/20 0.44
DRD1 P21728 1/20 0.43
TRPM8 Q7Z2W7 4/20 0.41
NPSR1 Q6W5P4 1/20 0.40
HHAT Q5VTY9 2/20 0.40
CYP2D6 P10635 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9508473 0.88 TRPM8 (0.45) ACEMTNR1BDRD1TRPM8NPSR1
SCHEMBL22366344 0.83 MTNR1B (0.48) ACEMTNR1BDRD1TRPM8NPSR1
SCHEMBL31020007 0.83 MTNR1B (0.48) ACEMTNR1BDRD1TRPM8NPSR1
SCHEMBL2138396 0.82 DRD1 (0.59) ACEMTNR1BDRD1NPSR1HHAT
SCHEMBL9508177 0.80 ACE (0.49) ACEMTNR1BDRD1TRPM8NPSR1
SCHEMBL9509872 0.78 MTNR1B (0.53) ACEMTNR1BDRD1NPSR1HHAT
SCHEMBL10770517 0.78 ACE (0.48) ACEMTNR1BDRD1TRPM8NPSR1
SCHEMBL9508456 0.77 HHAT (0.57) TRPM8HHATCYP2D6
SCHEMBL9508502 0.76 MTNR1B (0.57) ACEMTNR1BDRD1NPSR1HHAT
SCHEMBL9509163 0.76 MTNR1B (0.51) ACEMTNR1BDRD1NPSR1HHAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0230871-B1 HALOACYL 1-SUBSTITUTED-1,2,3,4-TETRAHYDROISOQUINOLINES AS HERBICIDE ANTIDOTES Monsanto Company (US) 1993-09-22 EP claimed
EP-0230871-A2 Haloacyl 1-substituted-1,2,3,4-tetrahydroisoquinolines as herbicide antidotes Monsanto Company (US) 1987-08-05 EP claimed
EP-0230871-B1 HALOACYL 1-SUBSTITUTED-1,2,3,4-TETRAHYDROISOQUINOLINES AS HERBICIDE ANTIDOTES Monsanto Company (US) 1993-09-22 EP disclosed
US-4755218-A Reducing acetochlor injury to corn by applying with antidote MONSANTO COMPANY (US) 1988-07-05 US disclosed
EP-0230871-A2 Haloacyl 1-substituted-1,2,3,4-tetrahydroisoquinolines as herbicide antidotes Monsanto Company (US) 1987-08-05 EP disclosed