SCHEMBL9517092

SCHEMBL9517092

COc1ccc(C(C)C(=O)NCCc2ccc(S(=O)(=O)NC(=O)c3ccc(CO)nc3)cc2)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.47
CA2 P00918 5/20 0.47
CA9 Q16790 5/20 0.47
CA12 O43570 4/20 0.47
CA4 P22748 4/20 0.47
TSHR P16473 1/20 0.47
ALDH1A1 P00352 3/20 0.45
CA7 P43166 1/20 0.44
CA14 Q9ULX7 1/20 0.44
QPCT Q16769 1/20 0.44
MAPT P10636 2/20 0.43
NLRP3 Q96P20 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
KMT2A Q03164 3/20 0.41
MEN1 O00255 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9516064 0.87 TSHR (0.62) CA1CA2CA9TSHRALDH1A1
SCHEMBL9516122 0.86 CA1 (0.62) CA1CA2CA9TSHRALDH1A1
SCHEMBL9517098 0.84 ALDH1A1 (0.61) CA1CA2CA9TSHRALDH1A1
SCHEMBL27535799 0.82 CA1 (0.47) CA1CA2CA9CA12CA4
SCHEMBL9517134 0.80 NLRP3 (0.68) TSHRALDH1A1MAPTNLRP3LMNA
SCHEMBL9515766 0.79 KMT2A (0.59) CA1CA2CA9CA12ALDH1A1
SCHEMBL9515821 0.79 POLB (0.49) CA1CA2CA9CA12TSHR
SCHEMBL9516791 0.78 LMNA (0.54) TSHRALDH1A1MAPTLMNATP53
SCHEMBL9519304 0.77 CA1 (0.55) CA1CA2CA9TSHRALDH1A1
SCHEMBL9518076 0.77 LMNA (0.44) CA1CA2CA9ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0567997-A1 4- or 5-(sulf)imido- and (sulfon)amidopyridines and their pyridine-N-oxides, process for their preparation and their use as pharmaceutical HOECHST AKTIENGESELLSCHAFT (DE) 1993-11-03 EP disclosed