SCHEMBL9517489

SCHEMBL9517489

O=C(c1ccc(F)c(F)c1)C(F)(Cl)Cl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.57
CES1 P23141 2/20 0.57
CHRNA1 P02708 1/20 0.44
CHRNG P07510 1/20 0.44
CHRNB1 P11230 1/20 0.44
CHRNB2 P17787 1/20 0.44
SLC6A2 P23975 1/20 0.44
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA4 P43681 1/20 0.44
SLC6A3 Q01959 1/20 0.44
CHRND Q07001 1/20 0.44
KCNQ3 O43525 4/20 0.41
KCNQ2 O43526 4/20 0.41
KCNQ5 Q9NR82 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KCNE1 P15382 1/20 0.40
KCNQ1 P51787 1/20 0.40
PLA2G7 Q13093 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9518686 0.86 CES2 (0.59) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL9517513 0.85 KCNQ3 (0.45) CES2CES1CHRNA3KCNQ3KCNQ2
SCHEMBL9516582 0.84 CES2 (0.57) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL15920928 0.83 CES1 (0.61) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL13543170 0.78 CES2 (0.59) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL9516563 0.74 CES1 (0.59) CES2CES1MEN1KMT2APLA2G7
SCHEMBL192962 0.74 CES2 (0.67) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL29470947 0.74 CES2 (0.67) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL29798141 0.73 CES1 (1.00) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL7967901 0.73 CES2 (0.73) CES2CES1CHRNA1CHRNGCHRNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105254519-B Synthesizing method of sitagliptin key intermediate 常州吉恩药业有限公司 2017-05-17 CN disclosed
EP-0411252-B1 Process for the preparation of fluorobenzoic acids RIEDEL DE HAEN AG (DE) 1993-11-03 EP disclosed
US-5093529-A Process for the preparation of fluorinated benzoic acids CASSELLA AKTIENGESELLSCHAFT (DE) 1992-03-03 US disclosed
EP-0411252-A1 Process for the preparation of fluorobenzoic acids RIEDEL-DE HAEN AKTIENGESELLSCHAFT (DE) 1991-02-06 EP disclosed