SCHEMBL9518482

SCHEMBL9518482

COC(=O)C(O)(O)CCC/C=C/c1c(-c2ccc(F)cc2)cn(C(C)C)c1C

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 7/20 0.49
ABCB1 P08183 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.30
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30
CACNA1G O43497 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9518969 0.81 HMGCR (0.52) HMGCRABCB1SLC6A4SLC6A3PTGDR2
SCHEMBL9518613 0.80 HMGCR (0.54) HMGCRSLC6A4SLC6A3
SCHEMBL10505092 0.79 HMGCR (0.52) HMGCRABCB1
SCHEMBL9023815 0.76 GCGR (0.31) HMGCR
SCHEMBL9024726 0.72 HMGCR (0.33) HMGCR
SCHEMBL9518404 0.72 HMGCR (0.65) HMGCR
SCHEMBL9750860 0.71 HMGCR (0.78) HMGCR
SCHEMBL9518535 0.71 HMGCR (0.54) HMGCRABCB1PTGDR2
SCHEMBL9750926 0.71 HMGCR (0.54) HMGCRABCB1PTGDR2
SCHEMBL9750845 0.70 HMGCR (0.56) HMGCRABCB1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0300249-B1 7-[1H-pyrrol-3-yl]-substituted 3,5-dihydroxy-heptane acids, their corresponding delta-lactones and salts, processes for their manufacture, their use as medicines, pharmaceutical preparations and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1993-02-03 EP disclosed
EP-0300249-A1 7-[1H-pyrrol-3-yl]-substituted 3,5-dihydroxy-heptane acids, their corresponding delta-lactones and salts, processes for their manufacture, their use as medicines, pharmaceutical preparations and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1989-01-25 EP disclosed