SCHEMBL9518937

SCHEMBL9518937

CC(C)(OC[C@@H]1C[C@H](S)CN1C(=O)OCc1ccc([N+](=O)[O-])cc1)C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
RAB9A P51151 2/20 0.38
HPGD P15428 1/20 0.38
NPC1 O15118 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CCR5 P51681 2/20 0.37
ATM Q13315 1/20 0.36
MAOB P27338 1/20 0.36
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9519806 0.87 ALDH1A1 (0.39) ALDH1A1MAPTRAB9AHPGDNPC1
SCHEMBL9520260 0.87 ALDH1A1 (0.36) ALDH1A1MAPTRAB9AHPGDNPC1
SCHEMBL10370916 0.86 RAB9A (0.42) ALDH1A1MAPTRAB9AHPGDNPC1
SCHEMBL9519722 0.86 CCR5 (0.38) ALDH1A1MAPTRAB9AHPGDNPC1
SCHEMBL10363296 0.84 MAOB (0.42) ALDH1A1MAPTRAB9AHPGDTDP1
SCHEMBL9519349 0.84 DPP8 (0.40) ALDH1A1MAPTHPGDTDP1CCR5
SCHEMBL9519480 0.83 RAB9A (0.40) ALDH1A1MAPTRAB9AHPGDNPC1
SCHEMBL10370030 0.83 RAB9A (0.42) ALDH1A1MAPTRAB9AHPGDNPC1
SCHEMBL7811546 0.83 RAB9A (0.43) ALDH1A1MAPTRAB9AHPGDNPC1
SCHEMBL9078142 0.83 HTT (0.40) ALDH1A1MAPTRAB9AHPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0280771-B1 3-Pyrrolidinylthio-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid derivatives and processes for the preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-07-28 EP disclosed
US-5061804-A 3-thiopyrrolidine as chemical intermediates FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-10-29 US disclosed
US-4963543-A BACTERICIDES, TREATING INFECTIOUS DISEASES; THIENAMYCINS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-10-16 US disclosed
EP-0280771-A1 3-Pyrrolidinylthio-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid derivatives and processes for the preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-09-07 EP disclosed