SCHEMBL9519841

SCHEMBL9519841

COc1cccc(/C(=C\C=C\CC(=O)O)c2ccccc2)c1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.55
MTNR1B P49286 5/20 0.55
GPR52 Q9Y2T5 1/20 0.49
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
CES2 O00748 1/20 0.49
CES1 P23141 1/20 0.49
MAOB P27338 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
PARP1 P09874 1/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
HSD11B1 P28845 1/20 0.46
BCHE P06276 2/20 0.45
HPGD P15428 1/20 0.45
ACHE P22303 1/20 0.45
KCNK3 O14649 1/20 0.45
KCNK9 Q9NPC2 1/20 0.45
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9522756 1.00 MTNR1A (0.55) MTNR1AMTNR1BGPR52NPC1RAB9A
SCHEMBL9519757 0.97 CES2 (0.51) MTNR1AMTNR1BGPR52NPC1RAB9A
SCHEMBL9519308 0.97 CES2 (0.51) MTNR1AMTNR1BGPR52NPC1RAB9A
SCHEMBL9520665 0.90 NPC1 (0.54) MTNR1AMTNR1BGPR52NPC1RAB9A
SCHEMBL9519518 0.90 NPC1 (0.54) MTNR1AMTNR1BGPR52NPC1RAB9A
SCHEMBL9522407 0.88 CES2 (0.53) GPR52NPC1RAB9ACES2CES1
SCHEMBL9523136 0.88 CES2 (0.53) GPR52NPC1RAB9ACES2CES1
SCHEMBL9521346 0.83 CA1 (0.49) GPR52NPC1RAB9ACES2CES1
SCHEMBL9521627 0.83 PAM (0.50) MTNR1AMTNR1BCES2CES1SMN1; SMN2
SCHEMBL9520140 0.83 PAM (0.50) MTNR1AMTNR1BCES2CES1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299379-B1 PENTADIENAMIDE PAF-ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
EP-0299379-A1 Pentadienamide PAF-antagonists F. HOFFMANN-LA ROCHE AG (CH) 1989-01-18 EP disclosed