Bicarbonate

Bicarbonate

SCHEMBL9520975

CC(C)=CC=C(c1ccccc1)c1ccccc1.O=C(O)O

nearest known ligand 0.47

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Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.47
MTNR1B P49286 1/20 0.47
CES2 O00748 4/20 0.46
CES1 P23141 4/20 0.46
ALDH1A1 P00352 3/20 0.42
TSHR P16473 3/20 0.42
DAO P14920 1/20 0.42
NAPRT Q6XQN6 1/20 0.42
TDP1 Q9NUW8 2/20 0.41
MAPK1 P28482 1/20 0.41
AKT1 P31749 1/20 0.40
CYP2C19 P33261 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
CYP1A2 P05177 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2C9 P11712 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MCOLN3 Q8TDD5 1/20 0.39
MAPT P10636 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44266 0.93 MTNR1A (0.42) MTNR1AMTNR1BCES2CES1ALDH1A1
SCHEMBL10397770 0.81 AKR1C3 (0.50) MTNR1AMTNR1BCES2CES1ALDH1A1
SCHEMBL10397769 0.81 AKR1C3 (0.50) MTNR1AMTNR1BCES2CES1ALDH1A1
SCHEMBL88322 0.81 ALDH1A1 (0.46) MTNR1AMTNR1BCES2CES1ALDH1A1
SCHEMBL183824 0.77 KDM1A (0.42) MTNR1AMTNR1BCES2CES1ALDH1A1
Bicarbonate SCHEMBL9521030 0.77 TSHR (0.43) MTNR1AMTNR1BCES2CES1ALDH1A1
Bicarbonate SCHEMBL9521636 0.77 TSHR (0.43) MTNR1AMTNR1BCES2CES1ALDH1A1
SCHEMBL19217672 0.77 CES2 (0.56) CES2CES1ALDH1A1TSHRDAO
Bicarbonate SCHEMBL9520143 0.77 TSHR (0.43) MTNR1AMTNR1BCES2CES1ALDH1A1
SCHEMBL9520971 0.76 MTNR1A (0.50) MTNR1AMTNR1BCES2CES1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299379-B1 PENTADIENAMIDE PAF-ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
EP-0299379-A1 Pentadienamide PAF-antagonists F. HOFFMANN-LA ROCHE AG (CH) 1989-01-18 EP disclosed