SCHEMBL9521709

SCHEMBL9521709

NC(=S)c1nc(-c2ccccc2)c[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
MAPT P10636 3/20 0.41
LMNA P02545 2/20 0.41
RAB9A P51151 1/20 0.38
ADORA2A P29274 3/20 0.37
ADORA1 P30542 2/20 0.37
MAP2K3 P46734 1/20 0.37
ASIC3 Q9UHC3 1/20 0.36
ATP4A P20648 1/20 0.36
ATP4B P51164 1/20 0.36
ASH1L Q9NR48 1/20 0.36
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
PDGFRB P09619 1/20 0.35
AGTR1 P30556 1/20 0.34
AURKA O14965 1/20 0.34
HSP90AA1 P07900 1/20 0.34
PRKACA P17612 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4243696 0.82 MAP2K3 (0.47) ALDH1A1MEN1KMT2AMAPTRAB9A
SCHEMBL21336547 0.82 MEN1 (0.38) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL7439224 0.79 ATP4A (0.37) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL9324010 0.78 TP53 (0.44) ALDH1A1MEN1KMT2ALMNARAB9A
SCHEMBL27662263 0.78 TP53 (0.41) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL14736658 0.77 ADORA3 (0.40) ALDH1A1MEN1KMT2AMAPTRAB9A
SCHEMBL2378994 0.75 ALDH1A1 (0.43) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL10622534 0.74 ALDH1A1 (0.45) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL14564382 0.73 DHODH (0.50) MAP2K3ASIC3AURKAPARP1
SCHEMBL7439221 0.72 MEN1 (0.35) ALDH1A1MEN1KMT2AMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1332952-C 4-substituted imidazole-2-thiones, 4-substituted imidazole-2-ones and related compounds and their use ALLERGAN INC (US) 2007-08-22 CN disclosed
CN-1671671-A 4- (substituted cycloalkylmethyl) imidazole-2-thiones, 4- (substituted cycloalkenylmethyl) imidazole-2-thiones, 4- (substituted cycloalkylmethyl) imidazol-2-ones, and 4- (substituted cycloalkenylmethyl) imidazol-2-ones, and related compounds ALLERGAN INC (US) 2005-09-21 CN disclosed
CN-1093535-C Imidazole derivative SHIONOGI & CO (JP) 2002-10-30 CN disclosed
CN-1158609-A Imidazole derivative SHIONOGI & CO (JP) 1997-09-03 CN disclosed
EP-0298196-B1 IMIDAZOLE COMPOUNDS AND BIOCIDAL COMPOSITIONS COMPRISING THE SAME ISHIHARA SANGYO KAISHA, LTD. (JP) 1993-06-02 EP disclosed
US-4995898-A Imidazole compounds and biocidal composition comprising the same for controlling harmful organisms ISHIHARA SANGYO KAISHA, LTD. (JP) 1991-02-26 US disclosed
EP-0298196-A1 Imidazole compounds and biocidal compositions comprising the same ISHIHARA SANGYO KAISHA, LTD. (JP) 1989-01-11 EP disclosed