SCHEMBL9521787

SCHEMBL9521787

O=C(Nc1ccccc1C(c1ccc(O)cc1)c1ccc(O)cc1)C12CC3CC(CC1C3)C2

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 7/20 0.43
CNR2 P34972 4/20 0.43
ADORA1 P30542 1/20 0.41
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
EPHX2 P34913 2/20 0.38
P2RX4 Q99571 1/20 0.38
ESR1 P03372 1/20 0.37
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9521389 0.87 CNR2 (0.57) P2RX7CNR2KMT2AALDH1A1GAA
SCHEMBL9521940 0.86 EPHX2 (0.42) P2RX7CNR2ADORA1KMT2AALDH1A1
SCHEMBL9520932 0.72 ALDH1A1 (0.49) P2RX7CNR2KMT2AALDH1A1GAA
SCHEMBL9124942 0.69 ALDH1A1 (0.59) P2RX7KMT2AALDH1A1GAATDP1
SCHEMBL9123251 0.69 GAA (0.62) KMT2AALDH1A1GAATDP1MAPT
SCHEMBL3685918 0.69 CNR2 (0.49) P2RX7CNR2ADORA1KMT2AALDH1A1
SCHEMBL9019625 0.69 KMT2A (0.36) P2RX7CNR2KMT2AALDH1A1GAA
SCHEMBL9124861 0.68 KMT2A (0.60) CNR2KMT2AALDH1A1GAATDP1
SCHEMBL9127786 0.68 KMT2A (0.49) KMT2AALDH1A1GAATDP1MEN1
SCHEMBL3805250 0.68 P2RX7 (0.56) P2RX7CNR2ADORA1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0395093-B1 TRIPHENYLMETHANE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-01 EP disclosed