SCHEMBL9523520

SCHEMBL9523520

CC1(C)C=C(c2ccncc2O)c2ccccc2O1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCNC P24863 15/20 0.40
CDK8 P49336 15/20 0.40
HASPIN Q8TF76 13/20 0.40
CDK19 Q9BWU1 7/20 0.35
KCNH2 Q12809 3/20 0.34
BACE1 P56817 1/20 0.34
OPRD1 P41143 2/20 0.34
CYP2D6 P10635 1/20 0.34
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
BUB1 O43683 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525775 0.79 RARA (0.41) CCNCCDK8HASPINCDK19
Hydrochloric Acid SCHEMBL9527636 0.78 RARA (0.40) CCNCCDK8HASPINCDK19
SCHEMBL9378940 0.76 SMN1; SMN2 (0.30) CCNCCDK8HASPINCDK19
SCHEMBL9525700 0.71 KDM4E (0.39) KCNH2OPRD1CYP2D6
SCHEMBL27313326 0.70 ALDH1A1 (0.37) KCNH2OPRD1
SCHEMBL9524666 0.68 METAP2 (0.37) KCNH2BACE1OPRD1
SCHEMBL769104 0.68 NISCH (0.40) KCNH2OPRD1CYP2D6
SCHEMBL12023184 0.68 IDO1 (0.48) CCNCCDK8HASPINMAOAMAOB
SCHEMBL9525977 0.67 OPRD1 (0.37) OPRD1
SCHEMBL12365910 0.67 RARA (0.51) KCNH2OPRD1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298452-B1 2H-1-BENZOPYRANE DERIVATIVES SUBSTITUTED IN POSITION 4 BY ARYL OR N-HETEROARYL F. HOFFMANN-LA ROCHE AG (CH) 1993-06-30 EP claimed
EP-0298452-B1 2H-1-BENZOPYRANE DERIVATIVES SUBSTITUTED IN POSITION 4 BY ARYL OR N-HETEROARYL F. HOFFMANN-LA ROCHE AG (CH) 1993-06-30 EP disclosed
US-5118694-A Hypotensive agents; treatment for cardiovascular and muscular disorders HOFFMANN-LA ROCHE INC. (US) 1992-06-02 US disclosed
US-4971982-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, SMOOTH MUSCLE DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-11-20 US disclosed
EP-0298452-A2 2H-1-benzopyrane derivatives substituted in position 4 by aryl or N-heteroaryl F. HOFFMANN-LA ROCHE AG (CH) 1989-01-11 EP disclosed