SCHEMBL9523934

SCHEMBL9523934

N#CC(C(=O)Nc1ccc(F)cc1)C(=O)c1nn(-c2ccccc2)c2c1CSc1ccc(NC(=O)C=O)cc1-2

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 10/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
RIPK1 Q13546 1/20 0.36
TP53 P04637 2/20 0.34
MAPT P10636 2/20 0.34
KCNJ6 P48051 2/20 0.34
KCNJ5 P48544 2/20 0.34
KCNJ3 P48549 2/20 0.34
PIK3CD O00329 2/20 0.33
PIK3R2 O00459 2/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
PIK3R5 Q8WYR1 2/20 0.33
PIK3R3 Q92569 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523480 0.96 MAPT (0.34) IKBKBALDH1A1LMNARIPK1TP53
SCHEMBL9523052 0.91 RIPK1 (0.37) IKBKBALDH1A1LMNARIPK1TP53
SCHEMBL9832532 0.89 ALDH1A1 (0.42) IKBKBALDH1A1LMNARIPK1TP53
SCHEMBL9525895 0.89 RIPK1 (0.38) IKBKBALDH1A1LMNARIPK1TP53
SCHEMBL9316088 0.88 TP53 (0.44) IKBKBALDH1A1LMNARIPK1TP53
SCHEMBL9525898 0.87 MAPT (0.40) IKBKBALDH1A1LMNARIPK1TP53
SCHEMBL9522542 0.87 TP53 (0.40) IKBKBALDH1A1LMNARIPK1TP53
SCHEMBL9837241 0.87 IKBKB (0.42) IKBKBALDH1A1LMNARIPK1
SCHEMBL9833948 0.87 ALDH1A1 (0.40) IKBKBALDH1A1LMNARIPK1TP53
SCHEMBL9522526 0.87 IKBKB (0.38) IKBKBALDH1A1LMNARIPK1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0420883-B1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
US-5166152-A Immunostimulants, bactericides, viricides, antitumor agents FARMITALIA CARLO ERBA S.R.L. (IT) 1992-11-24 US disclosed