SCHEMBL9525567

SCHEMBL9525567

CCC(=O)C(=O)Nc1ccc2c(c1)-c1c(c(C(=O)C(C#N)C(=O)Nc3cccc(C(F)(F)F)c3)nn1-c1ccccc1)CS2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNJ6 P48051 4/20 0.38
KCNJ5 P48544 4/20 0.38
KCNJ3 P48549 4/20 0.38
IDO1 P14902 1/20 0.38
POLB P06746 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
LMNA P02545 1/20 0.36
EPHX2 P34913 2/20 0.35
PTGS2 P35354 2/20 0.35
KLKB1 P03952 2/20 0.34
MAPT P10636 2/20 0.34
NR3C1 P04150 1/20 0.34
UBE2M P61081 1/20 0.34
DCUN1D1 Q96GG9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9316080 0.93 TP53 (0.37) LMNAMAPT
SCHEMBL9525574 0.92 LMNA (0.37) KCNJ6KCNJ5KCNJ3IDO1POLB
SCHEMBL9525895 0.91 RIPK1 (0.38) KCNJ6KCNJ5KCNJ3ALDH1A1LMNA
SCHEMBL9522374 0.90 RIPK1 (0.39) KCNJ6KCNJ5KCNJ3POLBMEN1
SCHEMBL9522526 0.90 IKBKB (0.38) ALDH1A1LMNAMAPT
SCHEMBL9316246 0.88 IDO1 (0.44) KCNJ6KCNJ5KCNJ3IDO1POLB
SCHEMBL9523720 0.88 MEN1 (0.37) MEN1ALDH1A1KMT2ASMN1; SMN2LMNA
SCHEMBL9831503 0.84 IDO1 (0.40) KCNJ6KCNJ5KCNJ3IDO1POLB
SCHEMBL9316085 0.84 MAPT (0.37) ALDH1A1KMT2ALMNAMAPT
SCHEMBL9525898 0.82 MAPT (0.40) KCNJ6KCNJ5KCNJ3ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0420883-B1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
US-5166152-A Immunostimulants, bactericides, viricides, antitumor agents FARMITALIA CARLO ERBA S.R.L. (IT) 1992-11-24 US disclosed
EP-0420883-A1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION. ERBA CARLO SPA (IT) 1991-04-10 EP disclosed
WO-1989012638-A1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-12-28 WO disclosed