SCHEMBL9525812

SCHEMBL9525812

Oc1ccnn1-c1c(Cl)cc(C(F)(F)F)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GABRA2 P47869 12/20 0.44
GABRB2 P47870 12/20 0.44
GABRB3 P28472 19/20 0.43
GABRP O00591 7/20 0.43
GABRD O14764 7/20 0.43
GABRA1 P14867 7/20 0.43
GABRB1 P18505 7/20 0.43
GABRG2 P18507 7/20 0.43
GABRA5 P31644 7/20 0.43
GABRA3 P34903 7/20 0.43
GABRA4 P48169 7/20 0.43
GABRE P78334 7/20 0.43
GABRA6 Q16445 7/20 0.43
GABRG1 Q8N1C3 7/20 0.43
GABRG3 Q99928 7/20 0.43
GABRQ Q9UN88 7/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9526822 0.87 GABRA2 (0.46) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL9458856 0.81 GABRB3 (0.54) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL10347986 0.81 GABRB3 (0.50) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL10437857 0.75 GABRB3 (0.46) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL9527645 0.74 BACE1 (0.42) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL10372959 0.73 BACE1 (0.43) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL10400984 0.73 GABRB3 (0.46) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL10556834 0.73 ACHE (0.41) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL20001726 0.73 HIF1A (0.41)
SCHEMBL10560567 0.72 SMN1; SMN2 (0.43) GABRA2GABRB2GABRB3GABRPGABRD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274642-B1 HERBICIDAL AND FUNGICIDAL AGENTS BASED ON SUBSTITUTED PYRAZOLIN-5-ONE DERIVATIVES BAYER AG (DE) 1993-08-11 EP disclosed
EP-0257296-B1 4-CYANO(NITRO)-5-OXY(THIO)-PYRAZOLE DERIVATIVES BAYER AG (DE) 1993-05-12 EP disclosed
US-5162528-A Pre- and post-emergence; phytaphthora in tomato plants; rice and wheat BAYER AKTIENGESELLSCHAFT (DE) 1992-11-10 US disclosed
US-5028717-A Herbicidal and fungicidal agents based on substituted pyrazolin-5-one derivatives BAYER AKTIENGESELLSCHAFT (DE) 1991-07-02 US disclosed
US-4909827-A Containing a C6-10 aryl group substituted in position 1 BAYER AKTIENGESELLSCHAFT (DE) 1990-03-20 US disclosed
US-4770692-A 4-cyano(nitro)-5-oxy(thio)-pyrazole derivatives, composition containing them, and herbicidal and plant growth regulating methods of using them BAYER AKTIENGESELLSCHAFT (DE) 1988-09-13 US disclosed
EP-0274642-A2 Herbicidal and fungicidal agents based on substituted pyrazolin-5-one derivatives BAYER AG (DE) 1988-07-20 EP disclosed
EP-0257296-A1 4-Cyano(nitro)-5-oxy(thio)-pyrazole derivatives BAYER AG (DE) 1988-03-02 EP disclosed
EP-0249033-A1 5-Oxy(thio)-pyrazole derivatives BAYER AG (DE) 1987-12-16 EP disclosed
US-4685956-A 1-aryl-5-hydrazino-pyrazoles, compositions containing them, and herbicidal method of using them BAYER AKTIENGESELLSCHAFT (DE) 1987-08-11 US disclosed
EP-0212353-A2 1-Aryl-5-hydrazino-pyrazoles BAYER AG (DE) 1987-03-04 EP disclosed