SCHEMBL9525819

SCHEMBL9525819

O=Cc1cccc2c1sc1ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.48
GPR3 P46089 1/20 0.48
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
LMNA P02545 1/20 0.44
THRB P10828 1/20 0.44
BLM P54132 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
PARP14 Q460N5 1/20 0.42
ALOX5 P09917 1/20 0.41
TNKS O95271 2/20 0.38
TNKS2 Q9H2K2 2/20 0.38
MAPT P10636 4/20 0.38
RAB9A P51151 2/20 0.38
ALDH1A1 P00352 2/20 0.38
TSHR P16473 1/20 0.38
TRIM24 O15164 1/20 0.38
TRIM33 Q9UPN9 1/20 0.38
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30705823 1.00 CYP2A6 (0.48) CYP2A6GPR3MEN1KMT2ALMNA
SCHEMBL19961736 0.86 PARP14 (0.51) CYP2A6GPR3MEN1KMT2ALMNA
SCHEMBL31689733 0.86 CYP2A6 (0.50) CYP2A6MEN1KMT2ALMNATHRB
SCHEMBL2786309 0.86 CYP2A6 (0.50) CYP2A6MEN1KMT2ALMNATHRB
SCHEMBL9540651 0.81 CYP2A6 (0.46) CYP2A6GPR3MEN1KMT2ALMNA
SCHEMBL9778942 0.81 CYP2A6 (0.49) CYP2A6MEN1KMT2ALMNATHRB
SCHEMBL17454809 0.81 GPR3 (0.48) CYP2A6GPR3MEN1KMT2ALMNA
SCHEMBL3057151 0.81 GPR3 (0.48) CYP2A6GPR3MEN1KMT2APARP14
SCHEMBL8149795 0.79 CYP2A6 (0.43) CYP2A6GPR3MEN1KMT2ALMNA
SCHEMBL25165131 0.78 GPR3 (0.45) GPR3MEN1KMT2ALMNAPARP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250189532-A1 1,6-DIYNE COMPOUND, ITS PREPARATION METHOD, AND PRODUCTS OBTAINED USING 1,6-DIYNE COMPOUND AS RAW MATERIAL AND THEIR APPLICATIONS FUJIAN INSTITUTE OF RESEARCH ON THE STRUCTURE OF MATTER, CHINESE ACADEMY OF SCIENCES (CN) 2025-06-12 US disclosed
CN-116730882-B Structure of 1, 6-diyne compound and application thereof 中国科学院福建物质结构研究所 2025-05-13 CN disclosed
EP-4488262-A1 1,6-DIYNE COMPOUND AND PREPARATION METHOD THEREFOR, AND PRODUCT OBTAINED USING 1,6-DIYNE COMPOUND AS RAW MATERIAL AND USE THEREOF Fujian Institute Of Research On The Structure Of Matter, Chinese Academy Of Sciences (CN) 2025-01-08 EP disclosed
WO-2024010732-A1 SMALL MOLECULE INHIBITORS OF GLUTAMINE TRANSPORTER ASCT2 AND METHODS OF USE THEREOF BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-01-11 WO disclosed
US-20230416422-A1 COMPOSITION, METHOD FOR MANUFACTURING SEMICONDUCTOR SUBSTRATE, POLYMER, AND METHOD FOR MANUFACTURING POLYMER JSR CORPORATION (JP) 2023-12-28 US disclosed
CN-116730882-A Structure of 1, 6-diyne compound and application thereof 中国科学院福建物质结构研究所 2023-09-12 CN disclosed
WO-2023165217-A1 1,6-DIYNE COMPOUND AND PREPARATION METHOD THEREFOR, AND PRODUCT OBTAINED USING 1,6-DIYNE COMPOUND AS RAW MATERIAL AND USE THEREOF 中国科学院福建物质结构研究所 2023-09-07 WO disclosed
US-20230192695-A1 THERMALLY ASSISTED DELAYED FLUORESCENT MATERIALS WITH TRIAD-TYPE MATERIALS UNIV ARIZONA STATE (US) 2023-06-22 US disclosed
US-20230192695-A1 THERMALLY ASSISTED DELAYED FLUORESCENT MATERIALS WITH TRIAD-TYPE MATERIALS UNIV ARIZONA STATE (US) 2023-06-22 US disclosed
CN-111763208-B Luminescent material and application thereof 北京鼎材科技有限公司 2023-04-07 CN disclosed
US-20150031686-A1 PHENYL-OXAZOLYL DERIVATIVES, PREPARATION METHOD THEREOF, AND RELATED APPLICATION OF THE PHENYL-OXAZOLYL DERIVATIVES AS AN IMPDH INHIBITOR INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2015-01-29 US disclosed
EP-0183439-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND USE AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-02-03 EP disclosed
US-5075455-A Microbiocides, antitumor agents BURROUGHS WELLCOME CO. (US) 1991-12-24 US disclosed
US-5049581-A Dibenzofurans having anti-tumor activity BURROUGHS WELLCOME CO. (US) 1991-09-17 US disclosed
US-5017600-A Antitumor BURROUGHS WELLCOME CO. (US) 1991-05-21 US disclosed
US-5008286-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-04-16 US disclosed
US-4970227-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1990-11-13 US disclosed
US-4965285-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-10-23 US disclosed
US-4866070-A ANTITUMOR AGENT BURROUGHS WELLCOME CO. (US) 1989-09-12 US disclosed
EP-0183439-A2 Polycyclic compounds, their preparation and use and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-06-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250189532-A1 1,6-DIYNE COMPOUND, ITS PREPARATION METHOD, AND PRODUCTS OBTAINED USING 1,6-DIYNE COMPOUND AS RAW MATERIAL AND THEIR APPLICATIONS HAO2, HAO1, TH CYP2A6 369/4885GPR3 737/4885MEN1 2755/4885
US-20230192695-A1 THERMALLY ASSISTED DELAYED FLUORESCENT MATERIALS WITH TRIAD-TYPE MATERIALS TTPA, TTC14, AAAS CYP2A6 3780/4885GPR3 4053/4885MEN1 2254/4885
US-20150031686-A1 PHENYL-OXAZOLYL DERIVATIVES, PREPARATION METHOD THEREOF, AND RELATED APPLICATION OF THE PHENYL-OXAZOLYL DERIVATIVES AS AN IMPDH INHIBITOR IMPDH1, IMPDH2, IMPA1 CYP2A6 668/4885GPR3 4502/4885MEN1 4023/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.