SCHEMBL952649

SCHEMBL952649

COc1cccc(-c2ccccc2CC#N)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.49
ABCB1 P08183 1/20 0.46
ABCC1 P33527 1/20 0.46
NAAA Q02083 1/20 0.44
ADORA2A P29274 2/20 0.44
ADORA1 P30542 2/20 0.44
ADORA2B P29275 1/20 0.44
BRD4 O60885 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CLK4 Q9HAZ1 2/20 0.43
LMNA P02545 2/20 0.43
MAPK1 P28482 2/20 0.43
TSHR P16473 1/20 0.43
PGR P06401 1/20 0.43
AR P10275 1/20 0.43
CYP1A1 P04798 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2085480 0.84 BACE1 (0.45) HTR7ARADRA2CCD274
SCHEMBL4665425 0.82 ABL1 (0.51) HTR7ABCB1CYP1A2CYP3A4CYP2C9
SCHEMBL8281062 0.81 HTR7 (0.52) HTR7ABCB1ABCC1BRD4CYP1A2
SCHEMBL8279410 0.81 MGAT2 (0.57) HTR7ABCB1ABCC1ADORA2AADORA1
SCHEMBL28854331 0.81 HTR7 (0.51) HTR7ABCB1ABCC1ADORA2AADORA1
SCHEMBL7704734 0.80 PTGER4 (0.50) NAAACYP4F2CYP4A11
Hydrochloric Acid SCHEMBL12490805 0.79 MGAT2 (0.56) HTR7ABCB1ABCC1ADORA2AADORA1
SCHEMBL2020140 0.79 ABL1 (0.59) ABCB1ADORA2AADORA1BRD4CYP1A2
SCHEMBL15456146 0.79 ADRA2C (0.45) HTR7ADORA2AADORA1ADORA2BCLK4
SCHEMBL1715907 0.78 IDO1 (0.54) HTR7ABCB1ABCC1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109222100-A A kind of ginseng Cordyceps militaris composition, ginseng Cordyceps militaris pressed candy and preparation method thereof 上海屹泽生物科技有限公司 2019-01-18 CN disclosed
EP-2121594-B1 QUATERNARY AMMONIUM DIPHENYLMETHYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE BIOPHARMA R & D IP LLC (US) 2015-10-21 EP disclosed
US-8802856-B2 Quaternary ammonium diphenylmethyl compounds useful as muscarinic receptor antagonists THERAVANCE BIOPHARMA R&D IP, LLC (US) 2014-08-12 US disclosed
US-20140051864-A1 QUATERNARY AMMONIUM DIPHENYLMETHYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2014-02-20 US disclosed
US-8592453-B2 Quaternary ammonium diphenylmethyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. (US) 2013-11-26 US disclosed
US-8378121-B2 Quaternary ammonium diphenylmethyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. (US) 2013-02-19 US disclosed
US-20110020231-A1 QUATERNARY AMMONIUM DIPHENYLMETHYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2011-01-27 US disclosed
US-20110021787-A1 QUATERNARY AMMONIUM DIPHENYLMETHYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2011-01-27 US disclosed
US-7834185-B2 Quaternary ammonium diphenylmethyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. (US) 2010-11-16 US disclosed
EP-2121594-A1 QUATERNARY AMMONIUM DIPHENYLMETHYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2009-11-25 EP disclosed
WO-2008103426-A1 QUATERNARY AMMONIUM DIPHENYLMETHYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2008-08-28 WO disclosed
US-20080207736-A1 Quaternary ammonium diphenylmethyl compounds useful as muscarinic receptor antagonists THERAVANCE BIOPHARMA R&D IP, LLC 2008-08-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080207736-A1 Quaternary ammonium diphenylmethyl compounds useful as muscarinic receptor antagonists CHRM2, CHRM5, CHRM1 HTR7 1175/4885ABCB1 969/4885ABCC1 926/4885
US-20110021787-A1 QUATERNARY AMMONIUM DIPHENYLMETHYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS CHRM2, CHRM5, CHRM1 HTR7 1175/4885ABCB1 969/4885ABCC1 926/4885
US-20110020231-A1 QUATERNARY AMMONIUM DIPHENYLMETHYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS CHRM2, CHRM5, CHRM1 HTR7 1175/4885ABCB1 969/4885ABCC1 926/4885
US-20140051864-A1 QUATERNARY AMMONIUM DIPHENYLMETHYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS CHRM2, CHRM5, CHRM1 HTR7 1175/4885ABCB1 969/4885ABCC1 926/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.