SCHEMBL9526679

SCHEMBL9526679

O=C(CBr)C1CCc2ccccc2C1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FAAH O00519 4/20 0.48
GHSR Q92847 1/20 0.47
MTNR1A P48039 4/20 0.45
MTNR1B P49286 4/20 0.45
P2RX7 Q99572 1/20 0.44
PLAU P00749 1/20 0.43
ANPEP P15144 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
F2 P00734 1/20 0.39
NPY5R Q15761 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5827457 0.87 FAAH (0.41) FAAHGHSRMTNR1AMTNR1BP2RX7
SCHEMBL8588823 0.83 MTNR1A (0.56) FAAHGHSRMTNR1AMTNR1BP2RX7
SCHEMBL6534265 0.81 GHSR (0.49) FAAHGHSRMTNR1AMTNR1BP2RX7
SCHEMBL11790481 0.80 MTNR1A (0.54) FAAHGHSRMTNR1AMTNR1BP2RX7
SCHEMBL6534185 0.78 FAAH (0.53) FAAHGHSRMTNR1AMTNR1BP2RX7
SCHEMBL6427539 0.78 FAAH (0.53) FAAHGHSRMTNR1AMTNR1BP2RX7
SCHEMBL5608206 0.78 FAAH (0.53) FAAHGHSRMTNR1AMTNR1BP2RX7
SCHEMBL367535 0.78 FAAH (0.53) FAAHGHSRMTNR1AMTNR1BP2RX7
SCHEMBL1193346 0.78 FAAH (0.53) FAAHGHSRMTNR1AMTNR1BP2RX7
SCHEMBL3195898 0.78 GHSR (0.49) FAAHGHSRMTNR1AMTNR1BP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0310745-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE ORION-YHTYMÄ OY (FI) 1993-01-27 EP disclosed
EP-0183492-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE Farmos-Yhtyma Oy (FI) 1989-11-15 EP disclosed
EP-0310745-A2 Substituted imidazole derivatives and their preparation and use ORION-YHTYMÄ OY (FI) 1989-04-12 EP disclosed
US-4689339-A 4-dihydroinden-2-yl-, 4-tetrahydronaphth-2-yl-, and 4-dihydrobenzofuran-2-ylimidazoles, useful to block α2 -adrenergic receptors FARMOS YHTYMA OY (FI) 1987-08-25 US disclosed
EP-0183492-A1 Substituted imidazole derivatives and their preparation and use Farmos-Yhtyma Oy (FI) 1986-06-04 EP disclosed