SCHEMBL9526882

SCHEMBL9526882

CCCOc1ccc(-c2ccc(C#N)c(=O)[nH]2)c(OCCC)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
KDM4E B2RXH2 4/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
GLA P06280 1/20 0.44
GAA P10253 1/20 0.44
MDM2 Q00987 3/20 0.39
XDH P47989 1/20 0.37
MAPK13 O15264 1/20 0.37
GCGR P47871 1/20 0.37
MAPK12 P53778 1/20 0.37
MAPK11 Q15759 1/20 0.37
MAPK14 Q16539 1/20 0.37
HPGD P15428 2/20 0.37
ACACB O00763 1/20 0.37
IDH1 O75874 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PDE3B Q13370 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7646373 0.93 L3MBTL1 (0.54) ALDH1A1KDM4EL3MBTL1GLAGAA
SCHEMBL9525981 0.93 KDM4E (0.48) ALDH1A1KDM4EL3MBTL1GLAGAA
SCHEMBL9702581 0.91 ALDH1A1 (0.44) ALDH1A1KDM4EL3MBTL1GLAGAA
SCHEMBL7646452 0.88 ALDH1A1 (0.42) ALDH1A1KDM4EL3MBTL1GLAGAA
SCHEMBL9525541 0.86 ALDH1A1 (0.52) ALDH1A1KDM4EL3MBTL1GLAGAA
SCHEMBL7645808 0.85 AR (0.40) ALDH1A1KDM4EL3MBTL1GLAGAA
SCHEMBL7409021 0.84 ALDH1A1 (0.39) ALDH1A1KDM4EL3MBTL1GLAGAA
SCHEMBL7644788 0.84 PDE5A (0.45) ALDH1A1KDM4EL3MBTL1GLAGAA
SCHEMBL7647544 0.84 ALDH1A1 (0.54) ALDH1A1KDM4EL3MBTL1GLAGAA
SCHEMBL7576593 0.83 ALDH1A1 (0.42) ALDH1A1KDM4EL3MBTL1GLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550576-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-07-14 EP disclosed
WO-1992006085-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-04-16 WO disclosed