SCHEMBL9527148

SCHEMBL9527148

CCc1nsc(OC(=O)Cl)c1C(=O)OC

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 4/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
LMNA P02545 3/20 0.32
HTT P42858 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PKM P14618 1/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9526569 0.88 LMNA (0.36) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL9446207 0.80 KDM4E (0.36) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL9446210 0.76 ALDH1A1 (0.40) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL9446238 0.73 LMNA (0.40) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL8550625 0.69 ABCC8 (0.34) TSHR
SCHEMBL9446209 0.69 LMNA (0.44) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL9526057 0.67 ACACB (0.31) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL11133645 0.62 PDE4D (0.51) KDM4ELMNAL3MBTL1MAPTKMT2A
SCHEMBL27193009 0.61 NPSR1 (0.36) ALDH1A1HPGDLMNAHTTL3MBTL1
SCHEMBL2901849 0.60

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337263-B1 ISOXAZOL(ISOTHIAZOLS)-5-CARBOXAMIDES BASF Aktiengesellschaft (DE) 1993-03-17 EP disclosed
EP-0337263-A2 Isoxazol(isothiazols)-5-carboxamides BASF Aktiengesellschaft (DE) 1989-10-18 EP disclosed