SCHEMBL9527561

SCHEMBL9527561

CC1(C)CC(c2ccccn2)c2cc(C(=O)c3ccccc3)ccc2O1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 2/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAPT P10636 1/20 0.38
ALDH1A1 P00352 2/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
AKR1C1 Q04828 1/20 0.36
BRD4 O60885 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
KMT2A Q03164 1/20 0.35
EZH2 Q15910 1/20 0.35
CNR2 P34972 2/20 0.35
ESR1 P03372 1/20 0.35
PABPC1 P11940 1/20 0.35
PLK1 P53350 1/20 0.35
HPGD P15428 1/20 0.34
CTNNB1 P35222 1/20 0.34
WNT3A P56704 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9628082 0.93 ABCC9 (0.34) ABCC9NPC1RAB9ANPSR1BRD4
SCHEMBL9524902 0.91 ESR1 (0.42) BRD4SMN1; SMN2KMT2AESR1PABPC1
SCHEMBL9628191 0.91 ABCC9 (0.33) ABCC9BRD4SMN1; SMN2KMT2AESR1
SCHEMBL9527983 0.90 TLR3 (0.40) NPC1RAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL9627698 0.87 BRD4 (0.37) NPSR1BRD4SMN1; SMN2ESR1PABPC1
SCHEMBL9524954 0.86 BRD4 (0.35) NPC1RAB9ANPSR1ALDH1A1BRD4
SCHEMBL9524371 0.86 KDM4E (0.42) NPC1RAB9ANPSR1MAPTALDH1A1
SCHEMBL9524908 0.84 MAPT (0.40) MAPTALDH1A1SMN1; SMN2KMT2AESR1
SCHEMBL9525760 0.79 TRPM5 (0.42) NPSR1SMN1; SMN2CNR2CNR1
SCHEMBL9524374 0.79 HTR2B (0.35) MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298452-B1 2H-1-BENZOPYRANE DERIVATIVES SUBSTITUTED IN POSITION 4 BY ARYL OR N-HETEROARYL F. HOFFMANN-LA ROCHE AG (CH) 1993-06-30 EP disclosed
US-5118694-A Hypotensive agents; treatment for cardiovascular and muscular disorders HOFFMANN-LA ROCHE INC. (US) 1992-06-02 US disclosed
US-4971982-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, SMOOTH MUSCLE DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-11-20 US disclosed
CN-1030582-A 1-benzopyran derivatives HOFFMANN LA ROCHE (CH) 1989-01-25 CN disclosed
EP-0298452-A2 2H-1-benzopyrane derivatives substituted in position 4 by aryl or N-heteroaryl F. HOFFMANN-LA ROCHE AG (CH) 1989-01-11 EP disclosed