SCHEMBL9627698

SCHEMBL9627698

CC1(C)CC(c2ccccn2)c2cc(C(=O)c3ccccc3I)ccc2O1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.33
CTNNB1 P35222 3/20 0.32
WNT3A P56704 1/20 0.32
TGFBR1 P36897 1/20 0.31
CTSD P07339 1/20 0.31
BACE1 P56817 1/20 0.31
TRPV1 Q8NER1 2/20 0.31
ESR1 P03372 1/20 0.31
PABPC1 P11940 1/20 0.31
PLK1 P53350 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TNKS O95271 3/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9628082 0.88 ABCC9 (0.34) BRD4SMN1; SMN2CTNNB1WNT3ATGFBR1
SCHEMBL9527561 0.87 ABCC9 (0.39) BRD4SMN1; SMN2CTNNB1WNT3AESR1
SCHEMBL9628191 0.86 ABCC9 (0.33) BRD4SMN1; SMN2CTNNB1WNT3ATGFBR1
SCHEMBL9524902 0.84 ESR1 (0.42) BRD4SMN1; SMN2CTNNB1WNT3ATGFBR1
SCHEMBL9527411 0.84 BRD4 (0.37) BRD4SMN1; SMN2CTNNB1WNT3ATRPV1
SCHEMBL9523546 0.83 TGFBR1 (0.39) BRD4SMN1; SMN2CTNNB1WNT3ATGFBR1
SCHEMBL9524954 0.82 BRD4 (0.35) BRD4SMN1; SMN2CTNNB1WNT3ATRPV1
SCHEMBL9524371 0.82 KDM4E (0.42) BRD4SMN1; SMN2NPSR1GAA
SCHEMBL9527983 0.82 TLR3 (0.40) SMN1; SMN2GAA
SCHEMBL9523970 0.79 DRD4 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5118694-A Hypotensive agents; treatment for cardiovascular and muscular disorders HOFFMANN-LA ROCHE INC. (US) 1992-06-02 US disclosed
US-4971982-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, SMOOTH MUSCLE DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-11-20 US disclosed