SCHEMBL9528261

SCHEMBL9528261

COc1cc(C(=O)O)ccc1C(C)c1c(Cl)[nH]c2ccc(CC3CCN(C)C3=O)cc12

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPN5 P54829 1/20 0.35
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 2/20 0.34
HPGD P15428 1/20 0.34
TLR9 Q9NR96 9/20 0.34
TLR8 Q9NR97 9/20 0.34
TLR7 Q9NYK1 9/20 0.34
KDM4E B2RXH2 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CNR1 P21554 1/20 0.32
ROCK2 O75116 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9528877 0.93 KMT2A (0.36) KMT2AALDH1A1MEN1HPGDTLR9
SCHEMBL9528727 0.85 CYSLTR2 (0.42) KMT2AMEN1CNR1
SCHEMBL9526764 0.85 NPC1 (0.37) KDM4EROCK2
SCHEMBL9531910 0.84 PLA2G4A (0.41) KMT2AMEN1CNR1
SCHEMBL9526686 0.78 NPC1 (0.36) ALDH1A1ROCK2
SCHEMBL9526859 0.78 B3GAT3 (0.36) HPGDROCK2
SCHEMBL9526830 0.76 NPC1 (0.35) ROCK2
SCHEMBL9490190 0.74 MAPT (0.41) PTPN5KMT2AALDH1A1MEN1TLR8
SCHEMBL9488311 0.74 ACACB (0.37) PTPN5HPGDTLR9TLR8TLR7
SCHEMBL9527469 0.74 NPC1 (0.35) KDM4EROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337767-B1 CYCLIC AMIDES ICI AMERICAS INC. (US) 1993-01-13 EP disclosed
US-5047402-A Leukotriene Antagonists ICI AMERICAS INC. (US) 1991-09-10 US disclosed
EP-0337767-A1 Cyclic amides ICI AMERICAS INC. (US) 1989-10-18 EP disclosed