SCHEMBL9524780

SCHEMBL9524780

O=C(CCN(C(=O)c1cncc(Br)c1)c1ccccc1)NCCNS(=O)(=O)c1cccc2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.39
P2RX7 Q99572 1/20 0.39
NPY5R Q15761 1/20 0.38
PRKCG P05129 4/20 0.38
PRKCZ Q05513 4/20 0.38
PRKCD Q05655 4/20 0.38
PRKD3 O94806 3/20 0.38
PRKCB P05771 3/20 0.38
PRKCA P17252 3/20 0.38
PRKCH P24723 3/20 0.38
PRKCI P41743 3/20 0.38
PRKCE Q02156 3/20 0.38
PRKCQ Q04759 3/20 0.38
PRKD1 Q15139 3/20 0.38
PRKACA P17612 3/20 0.38
PRKACG P22612 2/20 0.38
PRKACB P22694 2/20 0.38
EGFR P00533 1/20 0.38
MAPK1 P28482 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9528522 0.86 ALDH1A1 (0.45) SMN1; SMN2EGFRALDH1A1KDM4ENPC1
SCHEMBL9525975 0.85 SMN1; SMN2 (0.43) SMN1; SMN2MAPK1GLAALDH1A1LMNA
SCHEMBL9525948 0.84 PRKD3 (0.40) SMN1; SMN2P2RX7NPY5RPRKCGPRKCZ
Hydrochloric Acid SCHEMBL9526271 0.83 SLC6A9 (0.38) FLT3P2RX7NPY5RPRKCGPRKCZ
SCHEMBL9528510 0.83 SMN1; SMN2 (0.40) SMN1; SMN2ALDH1A1CYP1A2CYP2C19POLB
SCHEMBL9525116 0.81 SMN1; SMN2 (0.46) SMN1; SMN2EGFRMAPK1GLAALDH1A1
SCHEMBL9525362 0.80 BLM (0.43) SMN1; SMN2MAPK1CYP3A4CYP2D6ALDH1A1
SCHEMBL9525706 0.80 CYP1A2 (0.41) SMN1; SMN2ALDH1A1CYP1A2CYP2C19POLB
SCHEMBL9524974 0.79 ALDH1A1 (0.41) SMN1; SMN2MAPK1ALDH1A1HSD17B10LMNA
SCHEMBL9527984 0.79 SMN1; SMN2 (0.46) SMN1; SMN2EGFRMAPK1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed