SCHEMBL9699321

SCHEMBL9699321

CNCC1CN(N)c2ccccc2O1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.43
CA2 P00918 5/20 0.41
CASR P41180 3/20 0.41
ADRA2A P08913 1/20 0.40
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR7 P34969 1/20 0.40
ADRA1A P35348 1/20 0.40
HRH1 P35367 1/20 0.40
DRD3 P35462 1/20 0.40
HTR1A P08908 1/20 0.39
POLB P06746 1/20 0.38
ESR2 Q92731 1/20 0.38
MTNR1A P48039 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700481 0.80 CA2 (0.39) CA2ADRA2AHTR2AHTR2CADRA1A
SCHEMBL9532833 0.79 CASR (0.59) HTR6CASRADRA1AHTR1A
SCHEMBL9151791 0.79 HTR1A (0.40) CA2ADRA2AADRA1ADRD3HTR1A
SCHEMBL9701358 0.78 HTR6 (0.41) HTR6CA2CASRADRA2ADRD2
Hydrochloric Acid SCHEMBL9455227 0.78 CASR (0.58) HTR6CASRADRA1AHTR1A
SCHEMBL9153836 0.76 HTT (0.38) CA2ADRA2AADRA1ADRD3HTR1A
SCHEMBL11805714 0.76 GRM2 (0.51)
SCHEMBL9699225 0.76 HTR2A (0.42) CA2HTR2AHTR2CHRH1SIRT2
SCHEMBL9701550 0.74 ADRA2A (0.60) ADRA2ADRD2HTR2AHTR2CADRA1A
SCHEMBL9155416 0.74 HTT (0.46) POLBSIRT2SIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed